| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA921862 | B | Activity of human GRK5 kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
| 2. | ALA1057445 | B | Inhibition of GRK5 at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
| 3. | ALA1040650 | B | Residual activity of GRK5 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 4. | ALA1037597 | B | Residual activity of GRK5 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 5. | ALA1046822 | B | Residual activity of GRK5 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 6. | ALA1106959 | B | Inhibition of GRK5-mediated bovine tubulin phosphorylation by scintillation counting | 1 | ALA1154923 | single protein format | Scientific Literature | ||
| 7. | ALA1100484 | B | Inhibition of GRK5 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
| 8. | ALA1219848 | B | Inhibition of GRK5 ( assessed as residual activity at 1 uM ) | 2 | ALA1212910 | single protein format | Scientific Literature | ||
| 9. | ALA1219889 | B | Inhibition of human GRK5 | Homo sapiens | 2 | ALA1212911 | single protein format | Scientific Literature | |
| 10. | ALA1244441 | B | Inhibition of GRK5 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
| 11. | ALA1252430 | B | Inhibition of GRK5 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature | ||
| 12. | ALA1645976 | B | Inhibition of human GRK5 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature | |
| 13. | ALA1686356 | B | Inhibition of human GRK5 at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 14. | ALA1932867 | B | Inhibition of GRK5 | 2 | ALA1926590 | single protein format | Scientific Literature | ||
| 15. | ALA1963789 | F | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: GPRK5 | 346 | ALA1201862 | assay format | PubChem BioAssays | ||
| 16. | ALA2156648 | B | Inhibition of GRK5 at 1 uM | 1 | ALA2151019 | single protein format | Scientific Literature | ||
| 17. | ALA2219088 | B | Millipore: Percentage of residual kinase activity of GRK5 at 1uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | ALA2218924 | single protein format | Scientific Literature | |
| 18. | ALA2219089 | B | Millipore: Percentage of residual kinase activity of GRK5 at 10uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | ALA2218924 | single protein format | Scientific Literature | |
| 19. | ALA2343919 | B | Inhibition of GRK5 (unknown origin) | Homo sapiens | 1 | ALA2331117 | single protein format | Scientific Literature | |
| 20. | ALA2352892 | B | Inhibition of GRK5 (unknown origin) assessed as remaining activity at 10 uM relative to control | Homo sapiens | 2 | ALA2346597 | single protein format | Scientific Literature |
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