# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1292153 | Binding | Inhibition of human Nek3 | Homo sapiens | 1 | ALA1287713 | single protein format | Scientific Literature | |
2. | ALA1069800 | Binding | Residual activity of NEK3 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
3. | ALA1041158 | Binding | Residual activity of NEK3 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
4. | ALA1050311 | Binding | Residual activity of NEK3 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
5. | ALA1057497 | Binding | Inhibition of NEK3 at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
6. | ALA922011 | Binding | Activity of human NEK3 kinase at 1 uM | Homo sapiens | 1 | ALA1147076 | single protein format | Scientific Literature | |
7. | ALA941790 | Binding | Inhibition of NEK3 | 1 | ALA1140564 | single protein format | Scientific Literature | ||
8. | ALA1174942 | Binding | Inhibition of NEK3 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
9. | ALA1908567 | Binding | Binding constant for NEK3 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
10. | ALA4389369 | Binding | Inhibition of wild-type human full length NEK3 (M1 to R506 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
11. | ALA4389846 | Binding | Inhibition of wild-type human full length NEK3 (M1 to R506 residues) expressed in mammalian expression system at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
12. | ALA4382650 | Binding | Binding affinity to wild-type human full length NEK3 (M1 to R506 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature | |
13. | ALA1931517 | Binding | Inhibition of NEK3 | 2 | ALA1926590 | single protein format | Scientific Literature | ||
14. | ALA1646215 | Binding | Inhibition of human NEK3 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature | |
15. | ALA3241634 | Binding | Inhibition of human NEK3 assessed as enzyme activity at 1 uM relative to control | Homo sapiens | 1 | ALA3232845 | single protein format | Scientific Literature | |
16. | ALA4365857 | Binding | Inhibition of wild-type human full length NEK3 (M1 to R506 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
17. | ALA4366509 | Binding | Inhibition of human NEK3 at 100 nM using MBP as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature | |
18. | ALA4377735 | Binding | Inhibition of recombinant full-length human NEK3 at 1 uM using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 1 | ALA4376814 | single protein format | Scientific Literature | |
19. | ALA4378905 | Binding | Inhibition of recombinant human full length NEK3 at 10 uM using myelin basic protein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by scintillation counting method relative to control | Homo sapiens | 1 | ALA4376829 | single protein format | Scientific Literature | |
20. | ALA4379247 | Binding | Inhibition of recombinant full-length human NEK3 using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature |