| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2032527 | B | Inhibition of human histone demethylase LSD1 up to 100 uM | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 2. | ALA1798469 | B | Inhibition of partially purified LSD1 using histone H3K4Me2 peptide substrate by peroxidase-coupled assay | 3 | single protein format | Scientific Literature | |||
| 3. | ALA1798470 | B | Irreversible inhibition of partially purified LSD1 using histone H3K4Me2 peptide substrate by peroxidase-coupled assay | 2 | single protein format | Scientific Literature | |||
| 4. | ALA1798563 | B | Inhibition of LSD1 | 16 | single protein format | Scientific Literature | |||
| 5. | ALA1798564 | B | Ratio of Kinact to Ki for LSD1 | 2 | single protein format | Scientific Literature | |||
| 6. | ALA1798565 | B | Inhibition of GST-tagged LSD1 expressed in Escherichia coli | 2 | assay format | Scientific Literature | |||
| 7. | ALA1798573 | B | Reversible inhibition of LSD1 | 3 | single protein format | Scientific Literature | |||
| 8. | ALA1798574 | B | Inhibition of recombinant GST-tagged LSD1 expressed in baculovirus transfected Sf9 cells | 1 | cell-based format | Scientific Literature | |||
| 9. | ALA1798575 | B | Irreversible inhibition of LSD1 | 6 | single protein format | Scientific Literature | |||
| 10. | ALA1942527 | B | Inhibition of LSD1 | 14 | single protein format | Scientific Literature | |||
| 11. | ALA1942528 | B | Ratio of Kinact to Ki for LSD1 | 8 | single protein format | Scientific Literature | |||
| 12. | ALA1942546 | B | Inhibition of LSD1 at 10 uM | 1 | single protein format | Scientific Literature | |||
| 13. | ALA1799129 | B | Inhibition of human LSD1 | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 14. | ALA1799130 | B | Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as reduction of substrate turnover preincubated for 20 mins with substrate measured after 15 mins by mass spectrometric analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA1799131 | B | Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated for 20 mins with substrate measured after 30 mins by AmplexRed based fluorescence quenching assay | Homo sapiens | 11 | assay format | Scientific Literature | ||
| 16. | ALA1799132 | B | Inhibition of human truncated LSD1 lacking N-terminal 184 amino acids | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 17. | ALA926831 | B | Inhibition of human LSD1 | Homo sapiens | 7 | single protein format | Scientific Literature | ||
| 18. | ALA926833 | B | Ratio of Kinact to KI of human LSD1 | Homo sapiens | 7 | single protein format | Scientific Literature | ||
| 19. | ALA1025179 | B | Inhibition of LSD1 | 1 | single protein format | Scientific Literature | |||
| 20. | ALA1025180 | B | Inhibition of LSD1 at 1 uM | 1 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!