# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1932868 | B | Inhibition of GRK6 | 2 | single protein format | Scientific Literature | |||
2. | ALA1961880 | B | GSK_PKIS: GRK6 mean inhibition at 0.1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
3. | ALA1961881 | B | GSK_PKIS: GRK6 mean inhibition at 1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
4. | ALA2156649 | B | Inhibition of GRK6 at 1 uM | 1 | single protein format | Scientific Literature | |||
5. | ALA921863 | B | Activity of human GRK6 kinase at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
6. | ALA1057446 | B | Inhibition of GRK6 at 1 uM | 1 | single protein format | Scientific Literature | |||
7. | ALA1040651 | B | Residual activity of GRK6 at 0.1 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature | |||
8. | ALA1038408 | B | Residual activity of GRK6 at 1 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature | |||
9. | ALA1046823 | B | Residual activity of GRK6 at 10 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature | |||
10. | ALA1106960 | B | Inhibition of GRK6-mediated bovine tubulin phosphorylation by scintillation counting | 1 | single protein format | Scientific Literature | |||
11. | ALA1100485 | B | Inhibition of GRK6 at 10 uM | 2 | single protein format | Scientific Literature | |||
12. | ALA1244442 | B | Inhibition of GRK6 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | single protein format | Scientific Literature | |||
13. | ALA1252431 | B | Inhibition of GRK6 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | single protein format | Scientific Literature | |||
14. | ALA1645977 | B | Inhibition of human GRK6 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
15. | ALA2219090 | B | Millipore: Percentage of residual kinase activity of GRK6 at 1uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | single protein format | Scientific Literature | ||
16. | ALA2219091 | B | Millipore: Percentage of residual kinase activity of GRK6 at 10uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | single protein format | Scientific Literature | ||
17. | ALA2352891 | B | Inhibition of GRK6 (unknown origin) assessed as remaining activity at 10 uM relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
18. | ALA2352181 | B | Inhibition of GRK6 (unknown origin) using [gamma-33P]ATP assessed as residual activity at 3 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
19. | ALA2351969 | B | Inhibition of GRK6 (unknown origin) assessed as remaining activity at 1 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
20. | ALA2405115 | B | Inhibition of GRK6 (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature |