| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2071957 | B | Inhibition of KDM4C catalytic core-mediated demethylation of ARK(Me)3STGGK after 30 mins by FDH-coupled assay | Homo sapiens | 52 | single protein format | Scientific Literature | ||
| 2. | ALA2071958 | B | Inhibition of KDM4C catalytic core-mediated demethylation of ARK(Me)3STGGK at 500 uM after 30 mins by FDH-coupled assay in presence of increasing concentration of Fe(II) ions | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA2071960 | B | Inhibition of KDM4C | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA1942537 | B | Inhibition of KDM4C | 5 | single protein format | Scientific Literature | |||
| 5. | ALA1054733 | B | Inhibition of JMJD2C-mediated H3K36 demethylation in human 293T cells at 100 mM | 1 | cell-based format | Scientific Literature | |||
| 6. | ALA1054734 | B | Inhibition of JMJD2C-mediated H3K9 demethylation in human 293T cells at 100 mM | 1 | cell-based format | Scientific Literature | |||
| 7. | ALA1054737 | B | Inhibition of JMJD2C-mediated H3K9 demethylation activity at 3 mM | 5 | single protein format | Scientific Literature | |||
| 8. | ALA1055463 | B | Inhibition of JMJD2C-mediated H3K9 demethylation in human 293T cells at 2.5 mM | 2 | cell-based format | Scientific Literature | |||
| 9. | ALA1055464 | B | Inhibition of JMJD2C-mediated H3K36 demethylation in human 293T cells at 2.5 mM | 2 | cell-based format | Scientific Literature | |||
| 10. | ALA1055468 | B | Inhibition of JMJD2C-mediated H3K9 demethylation activity at 1 mM | 5 | single protein format | Scientific Literature | |||
| 11. | ALA1219074 | B | Inhibition of recombinant His-tagged JMJD2C expressed in Escherichia coli Rosetta 2 (DE3) pLysS cells by formaldehyde dehydrogenase-coupled assay | 15 | cell-based format | Scientific Literature | |||
| 12. | ALA1219079 | B | Ratio of compound IC50 to PCA IC50 for recombinant His-tagged JMJD2C | 1 | single protein format | Scientific Literature | |||
| 13. | ALA1219080 | B | Ratio of compound IC50 to NOG IC50 for recombinant His-tagged JMJD2C | 1 | single protein format | Scientific Literature | |||
| 14. | ALA1738633 | F | PUBCHEM_BIOASSAY: GASC-1 histone demethylase dose retest Measured in Cell-Free Homogeneous System Using Plate Reader - 2043-01_Inhibitor_Dose_CherryPick_Activity. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2123] | Homo sapiens | 150 | assay format | PubChem BioAssays | ||
| 15. | ALA2173246 | B | Inhibition of N-terminal GST-fused human JMJD2C catalytic domain amino acid 1 to 420 using H3K9me3 as substrate by mass spectrophotometric analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA2427610 | B | Inhibition of KDM4C (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assay | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 17. | ALA3110468 | B | Inhibition of recombinant JMJD2C (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen method | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 18. | ALA3390930 | B | Inhibition of GST-tagged human JMJD2C (1 to 420 residues) using H3K9me3 peptide as substrate expressed in Escherichia coli BL21 by MALDI-TOF/MS analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA3591677 | B | Inhibition of JMJD2C (unknown origin) using H3K9mel peptide | Homo sapiens | 17 | single protein format | Scientific Literature | ||
| 20. | ALA3624701 | B | Inhibition of KDM4C (unknown origin) using H3(1-21)K9Me3-GGK-biotin substrate incubated for 15 mins by alpha screen assay | Homo sapiens | 32 | single protein format | Scientific Literature |
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