| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1047550 | B | Inhibition of GLP | 1 | ALA1154694 | single protein format | Scientific Literature | ||
| 2. | ALA1047554 | B | Inhibition of GLP by Thioglo assay | 1 | ALA1154694 | single protein format | Scientific Literature | ||
| 3. | ALA1047555 | B | Inhibition of GLP by Alpha screen assay | 1 | ALA1154694 | single protein format | Scientific Literature | ||
| 4. | ALA1217454 | B | Activity at methyl transferase activity GLP by chemiluminescence based oxygen tunneling assay | 3 | ALA1212833 | single protein format | Scientific Literature | ||
| 5. | ALA1217457 | B | Activity at methyl transferase activity GLP by enzyme coupled S-adenocylehomocystein detection assay | 3 | ALA1212833 | single protein format | Scientific Literature | ||
| 6. | ALA1227298 | B | Inhibition of Histone H3 lysine 9 of GLP methyltransferase | 1 | ALA1221216 | single protein format | Scientific Literature | ||
| 7. | ALA1832316 | B | Inhibition of GLP assessed as hydrolysis of S-adenosyl-L-homocysteine after 2 mins by SAHH-coupled fluorescence assay | 1 | ALA1828613 | single protein format | Scientific Literature | ||
| 8. | ALA1832320 | B | Inhibition of GLP expressed in H1299 cells assessed as inhibition of dimethylation of p53 at lys 373 at 0.25 uM after 24 hrs by Western blot analysis | 1 | ALA1828613 | cell-based format | Scientific Literature | ||
| 9. | ALA2173362 | B | Competitive inhibition of GLP by fluorescence polarization assay in presence of fluorescein-labeled H3 peptide | 1 | ALA2169811 | single protein format | Scientific Literature | ||
| 10. | ALA2173366 | B | Binding affinity to human recombinant GLP catalytic domain amino acid 951 to 1235 expressed in Escherichia coli BL21 (DE3) by isothermal titration calorimetry assay | Homo sapiens | 1 | ALA2169811 | assay format | Scientific Literature | |
| 11. | ALA2173369 | B | Inhibition of human N-terminal hexahistidine-tagged GLP SET domain amino acid 951 to 1235 expressed in Escherichia coli BL21 (DE3) using Histone H3 peptide as substrate preincubated for 15 mins before substrate addition by mass spectrophotometric analysis | Homo sapiens | 1 | ALA2169811 | assay format | Scientific Literature | |
| 12. | ALA2330206 | B | Inhibition of GLP (unknown origin) using histone H3 (1 to 25) as substrate after 0.25 hrs by scintillation proximity assay in presence of [3H]-S-adenosylmethionine | Homo sapiens | 1 | ALA2321656 | single protein format | Scientific Literature | |
| 13. | ALA2350650 | B | Inhibition of EHMT1 (unknown origin) using [3H]SAM assessed as inhibition of biotinylated-H3 (1 to 25 amino acid residues) methylation at 0.1 to 100 uM after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA2346640 | single protein format | Scientific Literature | |
| 14. | ALA2443924 | B | Inhibition of lysine methyltransferase GLP (unknown origin) using [3H]-SAM as substrate after 0.25 hrs by scintillation proximity assay | Homo sapiens | 1 | ALA2440019 | single protein format | Scientific Literature | |
| 15. | ALA3111724 | B | Inhibition of GLP (unknown origin)-mediated incorporation of methyl group from [3H]-SAM into peptide substrate by scintillation proximity assay | Homo sapiens | 1 | ALA3108684 | single protein format | Scientific Literature | |
| 16. | ALA3129163 | B | Inhibition of human GLP (734 to 1235) using histone as substrate preincubated for 5 mins followed by substrate addition measured after 5 mins by liquid scintillation counting analysis in presence of [methyl-3H]-AdoMet | Homo sapiens | 6 | ALA3124813 | single protein format | Scientific Literature | |
| 17. | ALA3227364 | B | Inhibition of GLP (unknown origin) | Homo sapiens | 1 | ALA3217513 | single protein format | Scientific Literature | |
| 18. | ALA3266270 | B | Inhibition of methyltransferase activity of EHMT1 (unknown origin)-mediated dimethylation of a biotinylated histone H3 peptide at lysine-9 at 100 uM by FRET-based LANCE ultra G9a assay | Homo sapiens | 4 | ALA3259565 | single protein format | Scientific Literature | |
| 19. | ALA3266271 | B | Inhibition of methyltransferase activity of EHMT1 (unknown origin)-mediated dimethylation of a biotinylated histone H3 peptide at lysine-9 by FRET-based LANCE ultra G9a assay | Homo sapiens | 5 | ALA3259565 | single protein format | Scientific Literature | |
| 20. | ALA3266273 | B | Non-competitive inhibition of methyltransferase activity of EHMT1 (unknown origin) | Homo sapiens | 2 | ALA3259565 | single protein format | Scientific Literature |
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