# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1794385 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a: Hit Confirmation in b-rIgG Counterscreen. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504404] | 53 | assay format | PubChem BioAssays | |||
2. | ALA1804757 | B | Inhibition of G9a-mediated methylation of histone H3 at 100 uM after 90 mins by scintillation counting in presence of S-adenosyl-l-[methyl-3H]methionine | 3 | single protein format | Scientific Literature | |||
3. | ALA1832317 | B | Inhibition of G9a assessed as hydrolysis of S-adenosyl-L-homocysteine after 2 mins by SAHH-coupled fluorescence assay | 21 | single protein format | Scientific Literature | |||
4. | ALA1832319 | B | Inhibition of G9a expressed in H1299 cells assessed as inhibition of dimethylation of p53 at lys 373 at 0.25 uM after 24 hrs by Western blot analysis | 1 | cell-based format | Scientific Literature | |||
5. | ALA1832324 | B | Inhibition of G9a in human MDA-MB-231 cells assessed as reduction of H3K9me2 after 48 hrs by In-Cell Western assay | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
6. | ALA1832327 | B | Inhibition of G9a in human MCF7 cells assessed as reduction of H3K9me2 after 48 hrs by In-Cell Western assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
7. | ALA1832330 | B | Inhibition of G9a in human PC3 cells assessed as reduction of H3K9me2 after 48 hrs by In-Cell Western assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
8. | ALA1832333 | B | Inhibition of G9a in human 22Rv1 cells assessed as reduction of H3K9me2 after 48 hrs by In-Cell Western assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
9. | ALA1832435 | B | Inhibition of G9a in human HCT116 cells assessed as reduction of H3K9me2 after 48 hrs by In-Cell Western assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
10. | ALA1832438 | B | Inhibition of G9a in p53-deficient human HCT116 cells assessed as reduction of H3K9me2 after 48 hrs by In-Cell Western assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
11. | ALA1832441 | B | Inhibition of G9a in human IMR90 cells assessed as reduction of H3K9me2 after 48 hrs by In-Cell Western assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
12. | ALA1953573 | B | Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hr | 7 | single protein format | Scientific Literature | |||
13. | ALA1794504 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a: Hit Confirmation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504404] | 365 | assay format | PubChem BioAssays | |||
14. | ALA1798506 | B | Inhibition of lysine methyltransferase G9a | 3 | single protein format | Scientific Literature | |||
15. | ALA1046738 | B | Inhibition of G9a by Thioglo assay | 8 | single protein format | Scientific Literature | |||
16. | ALA1046739 | B | Inhibition of G9a at 1 uM by Thioglo assay | 6 | single protein format | Scientific Literature | |||
17. | ALA1046740 | B | Inhibition of G9a by Alpha screen assay | 13 | single protein format | Scientific Literature | |||
18. | ALA1047551 | B | Binding affinity to G9a by isothermal titration calorimetry | 1 | single protein format | Scientific Literature | |||
19. | ALA1047552 | B | Displacement of fluorescein [F-H391-150] peptide from G9a by fluorescence polarization assay | 1 | single protein format | Scientific Literature | |||
20. | ALA1047553 | B | Stabilization of G9a by differential scanning fluorimetry | 1 | single protein format | Scientific Literature |