# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3592286 | Binding | Inhibition of G9a (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | ALA3588844 | single protein format | Scientific Literature | |
2. | ALA3624015 | Binding | Inhibition of G9a (unknown origin) at 50 uM by scintillation proximity assay relative to control | Homo sapiens | 27 | ALA3621101 | single protein format | Scientific Literature | |
3. | ALA3624016 | Binding | Inhibition of G9a (unknown origin) at 10 uM by scintillation proximity assay relative to control | Homo sapiens | 27 | ALA3621101 | single protein format | Scientific Literature | |
4. | ALA3624017 | Binding | Inhibition of G9a (unknown origin) at 1 uM by scintillation proximity assay relative to control | Homo sapiens | 27 | ALA3621101 | single protein format | Scientific Literature | |
5. | ALA3624018 | Binding | Inhibition of G9a (unknown origin) using [histone H3 1 to 25 residues] and SAM substrate by scintillation proximity assay | Homo sapiens | 7 | ALA3621101 | single protein format | Scientific Literature | |
6. | ALA3626822 | Binding | Inhibition of G9a (unknown origin) at 100 uM preincubated for 15 mins followed by substrate addition measured after 60 mins by AlphaLISA method relative to control | Homo sapiens | 2 | ALA3621043 | single protein format | Scientific Literature | |
7. | ALA3784086 | Binding | Inhibition of human G9A at 10 and 50 uM | Homo sapiens | 1 | ALA3779843 | single protein format | Scientific Literature | |
8. | ALA3803123 | Binding | Inhibition of EHMT2 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA3797202 | single protein format | Scientific Literature | |
9. | ALA3812794 | Binding | Inhibition of G9a (unknown origin) by AlphaELISA | Homo sapiens | 1 | ALA3808369 | single protein format | Scientific Literature | |
10. | ALA3812795 | Binding | Inhibition of G9a (unknown origin) by ELISA | Homo sapiens | 1 | ALA3808369 | single protein format | Scientific Literature | |
11. | ALA3812796 | Binding | Inhibition of G9a (unknown origin) by fluorogenic assay | Homo sapiens | 1 | ALA3808369 | single protein format | Scientific Literature | |
12. | ALA3821561 | Binding | Inhibition of G9A (unknown origin) at 1 to 50 uM by scintillation proximity assay | Homo sapiens | 1 | ALA3817823 | single protein format | Scientific Literature | |
13. | ALA3825073 | Binding | Inhibition of G9a in human MCF7 nuclear extracts assessed as reduction in H3K9 levels at 15 uM after 48 hrs | Homo sapiens | 9 | ALA3822445 | cell-based format | Scientific Literature | |
14. | ALA3825074 | Binding | Inhibition of G9a in human MCF7 nuclear extracts assessed as reduction in H3K27 levels at 15 uM after 48 hrs | Homo sapiens | 8 | ALA3822445 | cell-based format | Scientific Literature | |
15. | ALA1217453 | Binding | Inhibition of methyl transferase activity of G9a assessed as inhibition of H3K9 methylation by chemiluminescence based oxygen tunneling assay | 37 | ALA1212833 | single protein format | Scientific Literature | ||
16. | ALA1217455 | Binding | Activity at methyl transferase activity G9a by enzyme coupled S-adenocylehomocystein detection assay | 25 | ALA1212833 | single protein format | Scientific Literature | ||
17. | ALA1217456 | Binding | Activity at methyl transferase activity G9a at 1 uM by enzyme coupled S-adenocylehomocystein detection assay | 12 | ALA1212833 | single protein format | Scientific Literature | ||
18. | ALA1217458 | Binding | Binding affinity to G9a by isothermal titration colorimetry | 2 | ALA1212833 | single protein format | Scientific Literature | ||
19. | ALA1227296 | Binding | Inhibition of recombinant G9a | 1 | ALA1221216 | single protein format | Scientific Literature | ||
20. | ALA1794385 | Functional | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a: Hit Confirmation in b-rIgG Counterscreen. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504404] | 53 | ALA1201862 | assay format | PubChem BioAssays |