| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1827278 | B | Activity of ERBB3 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
| 2. | ALA1908548 | B | Binding constant for ERBB3 kinase domain | 72 | single protein format | Scientific Literature | |||
| 3. | ALA930416 | B | Binding affinity to ErbB3 | 1 | single protein format | Scientific Literature | |||
| 4. | ALA1049971 | B | Binding affinity to ERBB3 assessed as percentage of kinase remaining bound to the bead at 1 uM by T7 phage display based binding assay | 1 | single protein format | Scientific Literature | |||
| 5. | ALA1169219 | B | Inhibition of ERBB3 at 1 uM | 6 | single protein format | Scientific Literature | |||
| 6. | ALA1174409 | B | Inhibition of ERBB3 at 10 uM | 2 | single protein format | Scientific Literature | |||
| 7. | ALA1244826 | B | Binding affinity to ERBB3 | 7 | single protein format | Scientific Literature | |||
| 8. | ALA2176625 | B | Inhibition of ERBB3 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
| 9. | ALA2214002 | B | Inhibition of ERBB3 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
| 10. | ALA2327210 | B | Inhibition of human recombinant HER-3 cytoplasmic domain (665 to 1339) autophosphorylation after 1 hr | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 11. | ALA2412603 | B | Inhibition of heregulin-stimulated HER3 phosphorylation in human MCF7 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA3088484 | B | Binding affinity to ERBB3 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA5250209 | B | Binding affinity to ERRB3 (unknown origin) assessed as strong interaction at 100 nM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA3112110 | B | Inhibition of ERBB3 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3749070 | B | Inhibition of ERBB3 (unknown origin) assessed as remaining activity at 1 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4025127 | B | Inhibition of wild-type human partial length ERBB3 (G684 to A987 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4034336 | B | Inhibition of ErbB3 Lysine 1 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4043938 | B | Inhibition of wild-type human partial length ERBB3 (G684 to A987 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA4048337 | B | Inhibition of partial length wild type human ERBB3 expressed in mammalian expression system at 0.5 uM by KINOMEscan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA4055198 | B | Inhibition of wild-type human partial length ERBB3 (G684 to A987 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature |
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