# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA942725 | B | Inhibition of AMPK | Homo sapiens | 1 | ALA1140564 | single protein format | Scientific Literature | |
2. | ALA948241 | B | Inhibition of AMPK at 10 uM | 6 | ALA1143190 | single protein format | Scientific Literature | ||
3. | ALA924594 | B | Inhibition of AMPK at 20 uM | 2 | ALA1144852 | single protein format | Scientific Literature | ||
4. | ALA1003321 | B | Inhibition of AMPK at 1 uM relative to control | 3 | ALA1136991 | single protein format | Scientific Literature | ||
5. | ALA994196 | B | Inhibition of AMPK | 1 | ALA1144228 | single protein format | Scientific Literature | ||
6. | ALA958269 | B | Inhibition of AMPK at 1 uM relative to control | 2 | ALA1150317 | single protein format | Scientific Literature | ||
7. | ALA1011054 | B | Inhibition of AMPKbeta1 at 100 nM relative to control | 1 | ALA1139385 | single protein format | Scientific Literature | ||
8. | ALA1012669 | B | Inhibition of AMPK at 5 uM | 2 | ALA1139352 | single protein format | Scientific Literature | ||
9. | ALA1047123 | B | Inhibition of human AMPK subunitB1 at 20 uM by FRET assay | Homo sapiens | 1 | ALA1156108 | single protein format | Scientific Literature | |
10. | ALA1259598 | B | Inhibition of AMPK at 1 uM | 1 | ALA1255571 | single protein format | Scientific Literature | ||
11. | ALA1285296 | B | Inhibition of AMPK at 0.1 uM | 1 | ALA1275361 | single protein format | Scientific Literature | ||
12. | ALA1806159 | B | Inhibition of AMPK assessed as residual enzyme activity at 10 uM | 1 | ALA1800061 | single protein format | Scientific Literature | ||
13. | ALA1941713 | B | Inhibition of AMPKbeta1 at 10 uM by colorimetric analysis | 4 | ALA1938312 | single protein format | Scientific Literature | ||
14. | ALA2019660 | B | Inhibition of AMPKB1 | 1 | ALA2016462 | single protein format | Scientific Literature | ||
15. | ALA2210936 | B | Inhibition of recombinant AMPK after 1 hr by scintillation counter analysis in presence of gamma-[33P]ATP | 1 | ALA2203238 | single protein format | Scientific Literature | ||
16. | ALA2343944 | B | Inhibition of AMPK (unknown origin) | Homo sapiens | 1 | ALA2331117 | single protein format | Scientific Literature | |
17. | ALA2390519 | B | Inhibition of AMPK (unknown origin) | Homo sapiens | 11 | ALA2384981 | single protein format | Scientific Literature | |
18. | ALA3707742 | B | Kinase Assay: Kinase assays were performed using the assay kit by Reaction Biology Corp (Malvern, Pa.). The compounds were tested at 10 concentrations by 3-fold serial dilutions starting at 30 μM. Staurosporin was used as a control nonspecific kinase inhibitor. In vitro kinase reactions using purified kinases were carried out in the presence of 10 μM ATP and test compounds. | Homo sapiens | 5 | ALA3639132 | single protein format | BindingDB Database | |
19. | ALA3859849 | B | Activation of human recombinant AMPK beta1 expressed in African green monkey COS7 cells or baculovirus infected insect cells assessed as increase in biotinylated AAC (1 to 120 residues) peptide phosphorylation at Ser-79 residue measured after 60 mins by Alphascreen assay | Homo sapiens | 1 | ALA3856285 | cell-based format | Scientific Literature | |
20. | ALA3859852 | B | Activation of AMPK beta1 in human HepG2 cells assessed as increase in phospho-ACC1 level at 1 uM after 2 hrs by ELISA relative to control | Homo sapiens | 1 | ALA3856285 | cell-based format | Scientific Literature |