# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1042727 | B | Inhibition of recombinant Taspase 1 assessed as accumulation of emitted fluorescence by FRET assay | 4 | single protein format | Scientific Literature | |||
2. | ALA1042728 | B | Inhibition of recombinant Taspase 1 assessed as accumulation of emitted fluorescence at 100 uM by FRET assay | 3 | single protein format | Scientific Literature | |||
3. | ALA1042729 | B | Inhibition of recombinant Taspase 1 assessed as loss of processing and accumulation of full length p45 fragment by radiographic in vitro cleavage assay added 30 mins before translated p45MLL | 4 | single protein format | Scientific Literature | |||
4. | ALA3992262 | B | Inhibition of recombinant Taspase1 (unknown origin) using [35S]-methionine labeled human MLL1 (2400-2900 residues) as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by SDS-PAGE based autoradiography | Homo sapiens | 4 | single protein format | Patent Bioactivity Data | ||
5. | ALA3992263 | B | Inhibition of recombinant Taspase1 (unknown origin) at 0.1 to 250 uM using [35S]-methionine labeled human MLL1 (2400-2900 residues) as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by SDS-PAGE based autoradiography | Homo sapiens | 1 | single protein format | Patent Bioactivity Data | ||
6. | ALA3992264 | B | Inhibition of recombinant Taspase1 (unknown origin) at 1 mM using [35S]-methionine labeled human MLL1 (2400-2900 residues) as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by SDS-PAGE based autoradiography | Homo sapiens | 1 | single protein format | Patent Bioactivity Data | ||
7. | ALA3992266 | B | Inhibition of recombinant Taspase1 (unknown origin) at 10 uM using [35S]-methionine labeled human MLL1 (2400-2900 residues) as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by SDS-PAGE based autoradiography | Homo sapiens | 1 | single protein format | Patent Bioactivity Data | ||
8. | ALA3992267 | B | Inhibition of recombinant Taspase1 (unknown origin) up to 0.1 mM using [35S]-methionine labeled human MLL1 (2400-2900 residues) as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by SDS-PAGE based autoradiography | Homo sapiens | 1 | single protein format | Patent Bioactivity Data | ||
9. | ALA3992268 | B | Covalent irreversible inhibition of recombinant Taspase1 (unknown origin) at 0.1 mM using [35S]-methionine labeled human MLL1 (2400-2900 residues) as substrate preincubated for 15 to 60 mins followed by substrate addition measured after 30 mins by SDS-PAGE based autoradiography | Homo sapiens | 1 | single protein format | Patent Bioactivity Data | ||
10. | ALA3992269 | B | Inhibition of recombinant Taspase1 (unknown origin) at 10 to 1000 uM using [35S]-methionine labeled human MLL1 (2400-2900 residues) as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by SDS-PAGE based autoradiography | Homo sapiens | 2 | single protein format | Patent Bioactivity Data | ||
11. | ALA3992273 | B | Non-competitive inhibition of recombinant Taspase1 (unknown origin) using FRPR as substrate preincubated with compound followed by substrate addition by fluorescence spectrometry | Homo sapiens | 1 | single protein format | Patent Bioactivity Data | ||
12. | ALA3992283 | B | Inhibition of recombinant Taspase1 (unknown origin) using FRPR as substrate preincubated with compound followed by substrate addition by fluorescence spectrometry | Homo sapiens | 7 | single protein format | Patent Bioactivity Data |