| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA865555 | B | Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cells | Rattus norvegicus | 19 | cell-based format | Scientific Literature | ||
| 2. | ALA865557 | B | Activity at chimeric rat/human MCH1R by accumulation of GTPgammaS | Rattus norvegicus | 2 | single protein format | Scientific Literature | ||
| 3. | ALA864915 | B | Inhibition of chimeric rat/human MCH1R at 10 uM | Rattus norvegicus | 2 | single protein format | Scientific Literature | ||
| 4. | ALA863646 | B | Inhibition of [125I]MCH binding to rat MCHR1 expressed in HEK293 cells by HT-SPA | Rattus norvegicus | 24 | cell-based format | Scientific Literature | ||
| 5. | ALA861266 | F | Activity at rat MCHR1 expressed in CHOK1-Gqi cells assessed as inhibition of MCH-induced calcium ion release by FLIPR assay | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA856556 | F | Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1 | Rattus norvegicus | 29 | cell-based format | Scientific Literature | ||
| 7. | ALA856558 | B | Displacement of 125I-[Phe13,Tyr19]-MCH from rat MCH-R1 | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 8. | ALA856559 | B | Inhibition of 125I-[Phe13,Tyr19]-MCH binding to rat MCH-R1 at 5uM | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 9. | ALA917759 | B | Binding affinity to rat MCH1 receptor | Rattus norvegicus | 14 | single protein format | Scientific Literature | ||
| 10. | ALA893404 | B | Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cells | Rattus norvegicus | 23 | cell-based format | Scientific Literature | ||
| 11. | ALA894439 | F | Antagonist activity at rat MCHR1 expressed in HEK293 cells assessed as effect on calcium mobilization | Rattus norvegicus | 22 | cell-based format | Scientific Literature | ||
| 12. | ALA894442 | B | Displacement of [3H]T-226296 from rat recombinant MCH1 receptor | Rattus norvegicus | 25 | single protein format | Scientific Literature | ||
| 13. | ALA894445 | F | Antagonist activity at rat MCH1 receptor expressed in HEK293 cells by FLIPR calcium mobility assay | Rattus norvegicus | 23 | cell-based format | Scientific Literature | ||
| 14. | ALA1039132 | B | Inhibition of rat MCH1R receptor | Rattus norvegicus | 2 | single protein format | Scientific Literature | ||
| 15. | ALA1821544 | B | Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation counting | Rattus norvegicus | 30 | cell-based format | Scientific Literature | ||
| 16. | ALA1821545 | F | Antagonist activity at rat MCHR1 expressed in CHO cells assessed as inhibition of MCH-induced GTPgammaS binding after 60 mins by scintillation counting | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA1833190 | B | Displacement of [125I]-S36057 from rat MCH1 receptor | Rattus norvegicus | 12 | single protein format | Scientific Literature | ||
| 18. | ALA1919497 | B | Displacement of [125I]-MCH(4-19) from rat MCHR1 expressed in CHO cells | Rattus norvegicus | 16 | cell-based format | Scientific Literature | ||
| 19. | ALA1924621 | F | Antagonist activity at rat MCHR1 expressed in HEK293 cells by aequorin bioluminescence assay | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA2032862 | F | Antagonist activity at rat MCHR1 assessed inhibition of MCH-mediated intracellular Ca2+ calcium mobilization | Rattus norvegicus | 1 | cell-based format | Scientific Literature |
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