# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1106961 | B | Inhibition of GRK7-mediated bovine tubulin phosphorylation by scintillation counting | 1 | ALA1154923 | single protein format | Scientific Literature | ||
2. | ALA1100486 | B | Inhibition of GRK7 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
3. | ALA1169251 | B | Inhibition of GRK7 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
4. | ALA1174442 | B | Inhibition of GRK7 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
5. | ALA1219789 | B | Inhibition of GRK7 at 1 uM by radiometric method | 2 | ALA1212904 | single protein format | Scientific Literature | ||
6. | ALA1244443 | B | Inhibition of GRK7 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
7. | ALA1244858 | B | Binding affinity to GRK7 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
8. | ALA1252432 | B | Inhibition of GRK7 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature | ||
9. | ALA1645978 | B | Inhibition of human GRK7 at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature | |
10. | ALA1826910 | B | Activity of GRK7 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
11. | ALA1908416 | B | Binding constant for GRK7 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
12. | ALA1961882 | B | GSK_PKIS: GRK7 mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
13. | ALA1961883 | B | GSK_PKIS: GRK7 mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
14. | ALA2156650 | B | Inhibition of GRK7 at 1 uM | 1 | ALA2151019 | single protein format | Scientific Literature | ||
15. | ALA2213531 | B | Inhibition of GRK7 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
16. | ALA2219092 | B | Millipore: Percentage of residual kinase activity of GRK7 at 1uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | ALA2218924 | single protein format | Scientific Literature | |
17. | ALA2219093 | B | Millipore: Percentage of residual kinase activity of GRK7 at 10uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | ALA2218924 | single protein format | Scientific Literature | |
18. | ALA2352890 | B | Inhibition of GRK7 (unknown origin) assessed as remaining activity at 10 uM relative to control | Homo sapiens | 2 | ALA2346597 | single protein format | Scientific Literature | |
19. | ALA2352180 | B | Inhibition of GRK7 (unknown origin) using [gamma-33P]ATP assessed as residual activity at 3 uM | Homo sapiens | 1 | ALA2346629 | single protein format | Scientific Literature | |
20. | ALA2351968 | B | Inhibition of GRK7 (unknown origin) assessed as remaining activity at 1 uM relative to control | Homo sapiens | 1 | ALA2346597 | single protein format | Scientific Literature |