# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1103982 | Binding | Activity of glucokinase assessed as stimulatory concentration required to increase 1.5 fold enzymatic activity | 58 | ALA1157747 | single protein format | Scientific Literature | ||
2. | ALA1103983 | Binding | Activity of glucokinase at 30 uM | 10 | ALA1157747 | single protein format | Scientific Literature | ||
3. | ALA1103984 | Binding | Activation of glucokinase at 1 uM measured per mg of protein | 2 | ALA1157747 | single protein format | Scientific Literature | ||
4. | ALA1103985 | Binding | Activation of glucokinase at 20 uM measured per mg of protein | 2 | ALA1157747 | single protein format | Scientific Literature | ||
5. | ALA1103986 | Binding | Activation of glucokinase assessed as increase in Vmax at 1 uM relative to control | 2 | ALA1157747 | single protein format | Scientific Literature | ||
6. | ALA1103987 | Binding | Activation of glucokinase at 20 uM relative to control | 2 | ALA1157747 | single protein format | Scientific Literature | ||
7. | ALA1103988 | Binding | Activation of glucokinase assessed as increase in Km at 1 uM relative to control | 2 | ALA1157747 | single protein format | Scientific Literature | ||
8. | ALA1103989 | Binding | Activation of glucokinase assessed as increase in Km at 20 uM relative to control | 2 | ALA1157747 | single protein format | Scientific Literature | ||
9. | ALA1103990 | Binding | Activity of glucokinase up to 10 uM | 2 | ALA1157747 | single protein format | Scientific Literature | ||
10. | ALA3240701 | Binding | Inhibition of biotin-tagged human GKRP/fluorescein-tagged GK interaction preincubated for 20 mins prior to GK addition measured after 2 to 4 hrs by AlphaScreen assay | Homo sapiens | 40 | ALA3232863 | single protein format | Scientific Literature | |
11. | ALA3131526 | Binding | Binding affinity to GKRP (unknown origin) by surface plasmon resonance analysis | Homo sapiens | 1 | ALA3124752 | single protein format | Scientific Literature | |
12. | ALA3131528 | Binding | Inhibition of biotin-tagged human GKRP-fluorescein-tagged human GK interaction preincubated for 20 mins followed by fluorescein-tagged human GK addition measured after 2 to 4 hrs by AlphaScreen assay | Homo sapiens | 24 | ALA3124752 | single protein format | Scientific Literature | |
13. | ALA3751185 | Binding | Binding affinity to human GKRP by surface plasmon resonance analysis | Homo sapiens | 14 | ALA3745641 | single protein format | Scientific Literature | |
14. | ALA3751192 | Binding | Binding affinity to human biotinylated AviTag GKRP assessed as inhibition of protein interaction with fluorescein tagged human glucokinase by AlphaScreen assay | Homo sapiens | 24 | ALA3745641 | single protein format | Scientific Literature | |
15. | ALA3751339 | Binding | Binding affinity to human GKRP assessed as inhibition of protein interaction with human glucokinase by measuring ATP depletion after 60 mins by luciferase-based luminescence assay | Homo sapiens | 1 | ALA3745641 | single protein format | Scientific Literature |