# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1116729 | B | Inhibition of NDR1 at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
2. | ALA1166588 | B | Inhibition of NDR1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
3. | ALA1174937 | B | Inhibition of NDR1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
4. | ALA1219263 | B | Inhibition of NDR1 at 3 uM | 1 | ALA1212924 | single protein format | Scientific Literature | ||
5. | ALA1244534 | B | Binding affinity to NDR1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
6. | ALA1827231 | B | Activity of NDR1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
7. | ALA1908764 | B | Binding constant for NDR1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
8. | ALA2015080 | B | Inhibition of NDR1 at 10 uM | 1 | ALA2010722 | single protein format | Scientific Literature | ||
9. | ALA2215437 | B | Inhibition of NDR1 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
10. | ALA3373410 | B | Inhibition of NDR1 (unknown origin) assessed as residual enzyme activity at 10 uM | Homo sapiens | 1 | ALA3352555 | single protein format | Scientific Literature | |
11. | ALA3430840 | B | Delta TM value showing the stabilisation of NDR1 produced by compound binding | Homo sapiens | 156 | ALA1145498 | single protein format | Scientific Literature | |
12. | ALA3631485 | B | Inhibition of STK38 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
13. | ALA3750171 | B | Inhibition of human STK38 using [KKRNRRLSVA] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
14. | ALA3991896 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 73 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
15. | ALA4025266 | B | Inhibition of wild-type human partial length NDR1 (N33 to E449 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
16. | ALA4034418 | B | Inhibition of NDR1 Lysine 1 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
17. | ALA4034419 | B | Inhibition of NDR1 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
18. | ALA4044077 | B | Inhibition of wild-type human partial length NDR1 (N33 to E449 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
19. | ALA4045770 | B | Inhibition of NDR1 conserved Lys1 (DTGHVYAMKILR) in human PBMC at 1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
20. | ALA4045771 | B | Inhibition of NDR1 conserved Lys2 (DIKPDNLLLDSK) in human PBMC at 1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature |