| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1067026 | B | Inhibition of human haspin at 0.1 uM | Homo sapiens | 1 | ALA1156855 | single protein format | Scientific Literature | |
| 2. | ALA1073724 | B | Inhibition of GSG2 at 3 to 6 uM relative to control | 1 | ALA1157712 | single protein format | Scientific Literature | ||
| 3. | ALA1102580 | B | Inhibition of GSG2 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
| 4. | ALA1114883 | B | Inhibition of Haspin at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
| 5. | ALA1103930 | B | Inhibition of haspin | 1 | ALA1157925 | single protein format | Scientific Literature | ||
| 6. | ALA1633357 | B | Inhibition of GSG2 at 10 uM | 1 | ALA1629532 | single protein format | Scientific Literature | ||
| 7. | ALA1645981 | B | Inhibition of human Haspin at 10 uM after 60 mins by TR-FRET assay | Homo sapiens | 1 | ALA1641539 | single protein format | Scientific Literature | |
| 8. | ALA1776212 | B | Inhibition of Haspin assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma counting | 1 | ALA1773059 | single protein format | Scientific Literature | ||
| 9. | ALA1947280 | B | Binding affinity to Haspin assessed as change in thermal denaturation at 10 uM by thermal stability shift assay | 16 | ALA1944596 | single protein format | Scientific Literature | ||
| 10. | ALA2014928 | B | Inhibition of Haspin at 10 uM | 1 | ALA2010722 | single protein format | Scientific Literature | ||
| 11. | ALA2015533 | B | Inhibition of human recombinant N-terminal MBP-tagged haspin kinase expressed in Escherichia coli DE3 at 10 uM after 10 mins by TR-FRET assay | Homo sapiens | 2 | ALA2010722 | assay format | Scientific Literature | |
| 12. | ALA2014113 | B | Inhibition of human recombinant N-terminal MBP-tagged haspin kinase expressed in Escherichia coli DE3 after 10 mins by TR-FRET assay | Homo sapiens | 20 | ALA2010722 | assay format | Scientific Literature | |
| 13. | ALA2156653 | B | Inhibition of Haspin at 1 uM | 1 | ALA2151019 | single protein format | Scientific Literature | ||
| 14. | ALA2184774 | B | Inhibition of haspin | 1 | ALA2176972 | single protein format | Scientific Literature | ||
| 15. | ALA2213528 | B | Inhibition of HASPIN assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 16. | ALA2219104 | B | Millipore: Percentage of residual kinase activity of GSG2 at 1uM relative to control. Control inhibitor: Staurosporine at 100.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | ALA2218924 | single protein format | Scientific Literature | |
| 17. | ALA2219105 | B | Millipore: Percentage of residual kinase activity of GSG2 at 10uM relative to control. Control inhibitor: Staurosporine at 100.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA | Homo sapiens | 158 | ALA2218924 | single protein format | Scientific Literature | |
| 18. | ALA2343916 | B | Inhibition of Haspin (unknown origin) | Homo sapiens | 1 | ALA2331117 | single protein format | Scientific Literature | |
| 19. | ALA2352550 | B | Inhibition of GSG2 (unknown origin) assessed as remaining activity at 10 uM relative to control | Homo sapiens | 1 | ALA2346597 | single protein format | Scientific Literature | |
| 20. | ALA2405113 | B | Inhibition of GSG2 (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | ALA2401733 | single protein format | Scientific Literature |
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