| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1040648 | B | Residual activity of GRK3 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 2. | ALA1037595 | B | Residual activity of GRK3 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 3. | ALA1046820 | B | Residual activity of GRK3 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
| 4. | ALA1106957 | B | Inhibition of GRK3-mediated bovine tubulin phosphorylation by scintillation counting | 1 | ALA1154923 | single protein format | Scientific Literature | ||
| 5. | ALA1102593 | B | Inhibition of GRK3 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
| 6. | ALA1243987 | B | Inhibition of GRK3 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
| 7. | ALA1251628 | B | Inhibition of ADRBK2 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature | ||
| 8. | ALA2156646 | B | Inhibition of GRK3 at 1 uM | 1 | ALA2151019 | single protein format | Scientific Literature | ||
| 9. | ALA2352894 | B | Inhibition of GRK3 (unknown origin) assessed as remaining activity at 10 uM relative to control | Homo sapiens | 2 | ALA2346597 | single protein format | Scientific Literature | |
| 10. | ALA2352184 | B | Inhibition of GRK3 (unknown origin) using [gamma-33P]ATP assessed as residual activity at 3 uM | Homo sapiens | 1 | ALA2346629 | single protein format | Scientific Literature | |
| 11. | ALA2351972 | B | Inhibition of GRK3 (unknown origin) assessed as remaining activity at 1 uM relative to control | Homo sapiens | 1 | ALA2346597 | single protein format | Scientific Literature | |
| 12. | ALA2406110 | B | Inhibition of ADRBK2 (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | ALA2401733 | single protein format | Scientific Literature | |
| 13. | ALA3630511 | B | Inhibition of GRK3 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 14. | ALA3734284 | B | Inhibition of GRK3 (unknown origin) after 90 to 120 mins by Kinase-Glo assay | Homo sapiens | 24 | ALA3727367 | single protein format | Patent Bioactivity Data | |
| 15. | ALA3751096 | B | Inhibition of GRK3 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3745631 | single protein format | Scientific Literature | |
| 16. | ALA3748201 | B | Inhibition of human GRK3 using casein as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
| 17. | ALA3762713 | B | Inhibition of GRK3 (unknown origin) at 100 nM | Homo sapiens | 1 | ALA3758169 | single protein format | Scientific Literature | |
| 18. | ALA3816348 | B | Inhibition of full length recombinant human GST-tagged GRK3 expressed in baculovirus expression system at 1 uM relative to control | Homo sapiens | 1 | ALA3813614 | assay format | Scientific Literature | |
| 19. | ALA3816686 | B | Inhibition of human GRK3 at 1 uM using casein as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
| 20. | ALA4025164 | B | Inhibition of wild-type human full length GRK3 (M1 to L688 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature |
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