# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2150703 | F | Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assay | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
2. | ALA2150705 | F | Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells at 10 mM after 20 mins by [35S]GTPgammaS binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
3. | ALA1105990 | B | Binding affinity to GPR81 | 4 | single protein format | Scientific Literature | |||
4. | ALA3300371 | F | Agonist activity at human HCA1 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation at 50 uM after 30 mins | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
5. | ALA3300372 | F | Agonist activity at human HCA1 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation up to 50 uM after 30 mins | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
6. | ALA3721244 | F | Agonist activity at human GPR81 expressed in CHO-K1 cell membranes pre-incubated for 5 to 10 mins before [35S]GTPgammaS addition followed by further incubation for 60 mins by microbeta counting based [35S]GTPgammaS binding assay | Homo sapiens | 142 | cell-based format | Patent Bioactivity Data | ||
7. | ALA3721245 | F | Agonist activity at human GPR81 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr by HTRF assay | Homo sapiens | 142 | cell-based format | Patent Bioactivity Data | ||
8. | ALA4611686 | F | Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production | Homo sapiens | 39 | cell-based format | Scientific Literature | ||
9. | ALA4611689 | F | Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production at 10 uM relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
10. | ALA4883488 | B | PRESTO-Tango GPCRome screening (HCA1) | 1 | single protein format | Donated Chemical Probes - SGC Frankfurt |