# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1815872 | B | Inhibition of human TRPM8 by fluorescent-based live-cell assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
2. | ALA1820170 | F | Agonist activity at human TRPM8 receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
3. | ALA1820171 | F | Antagonist activity at human TRPM8 receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
4. | ALA1958511 | F | Antagonist activity at human TRPM8 by calcium flux assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
5. | ALA1118224 | F | Antagonist activity at human TRPM8 channel | Homo sapiens | 1 | assay format | Scientific Literature | ||
6. | ALA1118250 | B | Activation of TRPM8 channel | 1 | single protein format | Scientific Literature | |||
7. | ALA1176441 | F | Antagonist activity at human TRPM8 receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
8. | ALA1224916 | F | Agonist activity at TRPM8 | 3 | assay format | Scientific Literature | |||
9. | ALA1243606 | B | Activity at human TRPM8 expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
10. | ALA1243607 | B | Activity at human TRPM8 R842A mutant expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
11. | ALA1243608 | B | Activity at human TRPM8 H845A mutant expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
12. | ALA1243609 | B | Activity at human TRPM8 R851Q mutant expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
13. | ALA1243610 | B | Activity at human TRPM8 K856A mutant expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
14. | ALA1243611 | B | Activity at human TRPM8 R862A mutant expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
15. | ALA1243612 | B | Activity at human TRPM8 R842K mutant expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
16. | ALA1243613 | B | Activity at human TRPM8 K856R mutant expressed in HEK293 cells assessed as compound concentration causing leftward shift of voltage for half maximal activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
17. | ALA1243614 | B | Binding affinity to human TRPM8 expressed in HEK293 cell membranes using [3H]labeled compound by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
18. | ALA1243615 | B | Displacement of [3H]menthol from human TRPM8 expressed in HEK293 cell membranes by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
19. | ALA1243616 | B | Displacement of [3H]menthol from human TRPM8 K856A mutant expressed in HEK293 cell membranes by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
20. | ALA1243617 | B | Displacement of [3H]menthol from human TRPM8 R842A mutant expressed in HEK293 cell membranes by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature |