# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA715019 | B | Compound was evaluated for inhibition of Staphylococcus aureus Methionine aminopeptidase 1 | Staphylococcus aureus | 3 | ALA1149091 | single protein format | Scientific Literature | |
2. | ALA715020 | B | Inhibitory activity against human methionine aminopeptidase-1 | 70 | ALA1146676 | single protein format | Scientific Literature | ||
3. | ALA716768 | B | Inhibitory activity against human methionine aminopeptidase-1; NT = Not tested | 29 | ALA1146676 | single protein format | Scientific Literature | ||
4. | ALA716769 | B | IInhibitory activity against Methionine aminopeptidase 1; ND = not determined | 1 | ALA1146714 | single protein format | Scientific Literature | ||
5. | ALA716770 | B | Inhibitory activity against Methionine aminopeptidase 1 | 4 | ALA1146714 | single protein format | Scientific Literature | ||
6. | ALA882587 | B | Inhibitory concentration against methionine aminopeptidase 1 | Homo sapiens | 1 | ALA1140404 | single protein format | Scientific Literature | |
7. | ALA853531 | B | Inhibition of MetAP1 | Homo sapiens | 1 | ALA1138906 | single protein format | Scientific Literature | |
8. | ALA894023 | B | Inhibition of human recombinant MetAP1 | Homo sapiens | 1 | ALA1148713 | single protein format | Scientific Literature | |
9. | ALA951176 | B | Inhibition of human methionine aminopeptidase 1 | Homo sapiens | 30 | ALA1143905 | single protein format | Scientific Literature | |
10. | ALA1027136 | B | Inhibition of methionine aminopeptidase 1 | 6 | ALA1152347 | single protein format | Scientific Literature | ||
11. | ALA1173890 | B | Inhibition of human MetAP1 at 25 uM | Homo sapiens | 52 | ALA1177825 | single protein format | Scientific Literature | |
12. | ALA1173891 | B | Inhibition of human MetAP1 | Homo sapiens | 26 | ALA1177825 | single protein format | Scientific Literature | |
13. | ALA2187527 | B | Inhibition of Mn(II) form of human methionine aminopeptidase1 expressed in Escherichia coli at 100 mM | Homo sapiens | 4 | ALA2177059 | assay format | Scientific Literature | |
14. | ALA2339332 | B | Inhibition of human MetAP1 expressed in Escherichia coli BL21(lambdaDE3) using Met-AMC as substrate at 10 uM incubated for 30 mins prior to substrate addition measured for 15 mins fluorometric analysis | Homo sapiens | 7 | ALA2331445 | assay format | Scientific Literature | |
15. | ALA2378642 | B | Inhibition of methionine aminopeptidase 1 in HEK293 cells expressing 3xFLAG-tagged BTF3 assessed as increase in [35S]-Met in solution at 10 uM after 30 mins by scintillation counting analysis | Homo sapiens | 1 | ALA2375230 | cell-based format | Scientific Literature | |
16. | ALA2378643 | B | Inhibition of methionine aminopeptidase 1 in HEK293 cells expressing 3xFLAG-tagged BTF3 assessed as increase in [35S]-Met in solution at 100 nM after 30 mins by scintillation counting analysis | Homo sapiens | 1 | ALA2375230 | cell-based format | Scientific Literature | |
17. | ALA2378644 | B | Inhibition of methionine aminopeptidase 1 in HEK293 cells expressing 3xFLAG-tagged TXNL1 assessed as increase in [35S]-Met in solution at 10 uM after 30 mins by scintillation counting analysis relative to control | Homo sapiens | 1 | ALA2375230 | cell-based format | Scientific Literature | |
18. | ALA2378645 | B | Inhibition of human methionine aminopeptidase 1 up to 250 uM | Homo sapiens | 1 | ALA2375230 | single protein format | Scientific Literature | |
19. | ALA2378646 | B | Inhibition of human methionine aminopeptidase 1 at 100 uM relative to control | Homo sapiens | 3 | ALA2375230 | single protein format | Scientific Literature | |
20. | ALA2378687 | B | Inhibition of methionine aminopeptidase 1 in HDFa cells assessed as increase in ratio of unprocessed 14-3-3gamma to total 14-3-3gamma at 250 uM after 24 hrs by immunoblotting analysis relative to DMSO-treated control | Homo sapiens | 1 | ALA2375230 | cell-based format | Scientific Literature |