# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA760612 | B | Inhibition of [3H]- (+) - pentazocine binding to PCP receptor obtained from tissue homogenate preparation of fresh whole rat brain minus cerebellum | Rattus norvegicus | 1 | ALA1131468 | tissue-based format | Scientific Literature | |
2. | ALA760613 | B | Inhibition of [3H]-TCP binding to PCP receptor obtained from tissue homogenate preparation of fresh whole rat brain minus cerebellum | Rattus norvegicus | 5 | ALA1131468 | tissue-based format | Scientific Literature | |
3. | ALA760614 | B | Inhibition of binding to PCP receptor obtained from tissue homogenate preparation of fresh whole rat brain minus cerebellum | Rattus norvegicus | 2 | ALA1131468 | tissue-based format | Scientific Literature | |
4. | ALA873407 | B | Compound was tested for its binding affinity towards PCP receptor using [3H](+)-NANM in the presence of 5 uM haloperidol from rat brain | Rattus norvegicus | 1 | ALA1131209 | assay format | Scientific Literature | |
5. | ALA760615 | B | Inhibition of [3H]- (+) - pentazocine binding to PCP receptor obtained from tissue homogenate preparation of fresh whole rat brain minus cerebellum | Rattus norvegicus | 1 | ALA1131468 | tissue-based format | Scientific Literature | |
6. | ALA759461 | B | Ratio of binding towards PCP receptor to that of sigma receptor | Rattus norvegicus | 5 | ALA1131468 | single protein format | Scientific Literature | |
7. | ALA759462 | B | Potency for binding towards PCP receptor relative to that of phencyclidine | Rattus norvegicus | 7 | ALA1131468 | single protein format | Scientific Literature | |
8. | ALA764432 | B | Inhibition of [3H]1-[1-(2-thienyl) piperidine ([3H]TCP) binding to phencyclidine receptor | Rattus norvegicus | 26 | ALA1124619 | single protein format | Scientific Literature | |
9. | ALA1110131 | B | Inhibition of carboxypeptidase P | 1 | ALA1157839 | single protein format | Scientific Literature | ||
10. | ALA1261609 | B | Inhibition of human PrCP by FRET | Homo sapiens | 62 | ALA1255224 | single protein format | Scientific Literature | |
11. | ALA1261610 | B | Inhibition of human PrCP at 5 uM by FRET | Homo sapiens | 22 | ALA1255224 | single protein format | Scientific Literature | |
12. | ALA1261611 | B | Inhibition of human PrCP by FRET in presence of 1% mouse serum albumin | Homo sapiens | 18 | ALA1255224 | single protein format | Scientific Literature | |
13. | ALA1687133 | B | Inhibition of human PrCP | Homo sapiens | 33 | ALA1681696 | single protein format | Scientific Literature | |
14. | ALA1687190 | B | Inhibition of human PrCP at 5 uM | Homo sapiens | 1 | ALA1681696 | single protein format | Scientific Literature | |
15. | ALA1942257 | B | Inhibition of recombinant human PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate measured for 30 mins by continuous fluorometric assay | Homo sapiens | 46 | ALA1938250 | single protein format | Scientific Literature | |
16. | ALA1941295 | B | Inhibition of recombinant human PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate at 10 uM measured for 30 mins by continuous fluorometric assay | Homo sapiens | 1 | ALA1938250 | single protein format | Scientific Literature | |
17. | ALA1953699 | B | Inhibition of human PrCP | Homo sapiens | 24 | ALA1949630 | single protein format | Scientific Literature | |
18. | ALA1953317 | B | Inhibition of human recombinant PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate after 30 mins by fluorescence analysis | Homo sapiens | 37 | ALA1949605 | single protein format | Scientific Literature | |
19. | ALA1953320 | B | Inhibition of human recombinant PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate at 5 uM after 30 mins by fluorescence analysis | Homo sapiens | 1 | ALA1949605 | single protein format | Scientific Literature | |
20. | ALA1955691 | B | Inhibition of human recombinant PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate at 5 uM for 30 mins by continuous fluorimetric assay | Homo sapiens | 3 | ALA1949559 | single protein format | Scientific Literature |