# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1826212 | B | Activity of MAK kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
2. | ALA1166054 | B | Inhibition of MAK at 1 uM | 6 | single protein format | Scientific Literature | |||
3. | ALA1174887 | B | Inhibition of MAK at 10 uM | 2 | single protein format | Scientific Literature | |||
4. | ALA1244488 | B | Binding affinity to MAK | 7 | single protein format | Scientific Literature | |||
5. | ALA1908722 | B | Binding constant for MAK kinase domain | 72 | single protein format | Scientific Literature | |||
6. | ALA2210637 | B | Inhibition of MAK assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
7. | ALA2342047 | B | Inhibition of MAK (unknown origin) assessed as residual activity at 100 nM after 1 hr by competitive binding assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA3624242 | B | Inhibition of MAK (unknown origin) at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
9. | ALA4025216 | B | Inhibition of wild-type human partial length MAK (M1 to P314 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
10. | ALA4044027 | B | Inhibition of wild-type human partial length MAK (M1 to P314 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
11. | ALA4055209 | B | Inhibition of wild-type human partial length MAK (M1 to P314 residues) expressed in bacterial expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
12. | ALA4157106 | B | Binding affinity to wild-type human partial length MAK (M1 to P314 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
13. | ALA4185885 | B | Binding affinity to wild-type human partial length MAK (M1 to P314 residues) expressed in Escherichia coli BL21 at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
14. | ALA4191032 | B | Inhibition of recombinant full-length human MAK at 1 uM using RRRFRPASPLRGPPK as substrate after 120 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
15. | ALA4230785 | B | Binding affinity to wild-type human partial length MAK (M1 to P314 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
16. | ALA4264374 | B | Binding affinity to wild-type human partial length MAK (M1 to P314 residues) expressed in bacterial expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
17. | ALA4307884 | B | Binding affinity to wild-type human partial length MAK (M1 to P314 residues) expressed in bacterial expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
18. | ALA4314868 | B | Inhibition of recombinant full-length human MAK assessed as residual activity at 10 uM using RRRFRPASPLRGPPK as substrate measured after 120 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
19. | ALA4327751 | B | Inhibition of human MAK assessed as residual activity at 1 uM using MBP as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
20. | ALA4328115 | B | Inhibition of human MAK assessed as residual activity at 100 uM using MBP as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature |