# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1167713 | B | Inhibition of STK39 at 1 uM | 7 | ALA1165965 | single protein format | Scientific Literature | ||
2. | ALA1175027 | B | Inhibition of STK39 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
3. | ALA1244991 | B | Binding affinity to STK39 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
4. | ALA1827259 | B | Activity of STK39 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
5. | ALA1908768 | B | Binding constant for STK39 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
6. | ALA2209685 | B | Inhibition of STK39 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
7. | ALA3631487 | B | Inhibition of STK39 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
8. | ALA3750173 | B | Inhibition of human STK39 using MBP substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
9. | ALA3816855 | B | Inhibition of human STK39 at 1 uM using MBP substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
10. | ALA4025400 | B | Inhibition of wild-type human partial length STK39 (P43 to I357 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
11. | ALA4034496 | B | Inhibition of STLK3 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
12. | ALA4044211 | B | Inhibition of wild-type human partial length STK39 (P43 to I357 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
13. | ALA4045841 | B | Inhibition of STLK3 conserved Lys2 (DLKAGNILLGEDGSVQIADFGVSAFLATGGDVTR) in human PBMC at 1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
14. | ALA4046082 | B | Inhibition of STLK3 conserved Lys2 (DLKAGNILLGEDGSVQIADFGVSAFLATGGDVTR) in human PBMC at 0.1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
15. | ALA4055263 | B | Inhibition of wild-type human partial length STLK3 (P43 to I357 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
16. | ALA4151508 | B | Inhibition of N-terminal His tagged recombinant full-length human STK39 expressed in baculovirus infected Sf9 cells at 1 uM | Homo sapiens | 1 | ALA4145674 | cell-based format | Scientific Literature | |
17. | ALA4157290 | B | Binding affinity to wild-type human partial length STK39 (P43 to I357 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
18. | ALA4186069 | B | Binding affinity to wild-type human partial length STK39 (P43 to I357 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | cell-based format | Scientific Literature | |
19. | ALA4230969 | B | Binding affinity to wild-type human partial length STK39 (P43 to I357 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
20. | ALA4264558 | B | Binding affinity to wild-type human partial length STK39 (P43 to I357 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature |