| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1827759 | B | Activity of CDKL3 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
| 2. | ALA1908519 | B | Binding constant for CDKL3 kinase domain | 72 | single protein format | Scientific Literature | |||
| 3. | ALA1168827 | B | Inhibition of CDKL3 at 1 uM | 6 | single protein format | Scientific Literature | |||
| 4. | ALA1174172 | B | Inhibition of CDKL3 at 10 uM | 2 | single protein format | Scientific Literature | |||
| 5. | ALA1244765 | B | Binding affinity to CDKL3 | 7 | single protein format | Scientific Literature | |||
| 6. | ALA2209328 | B | Inhibition of CDKL3 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
| 7. | ALA3112115 | B | Inhibition of CDKL3 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4025062 | B | Inhibition of wild-type human partial length CDKL3 (M1 to D327 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA4043873 | B | Inhibition of wild-type human partial length CDKL3 (M1 to D327 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA4055166 | B | Inhibition of wild-type human partial length CDKL3 (M1 to D327 residues) expressed in bacterial expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 11. | ALA4156952 | B | Binding affinity to wild-type human partial length CDKL3 (M1 to D327 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA4185731 | B | Binding affinity to wild-type human partial length CDKL3 (M1 to D327 residues) expressed in Escherichia coli BL21 at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 13. | ALA4230631 | B | Binding affinity to wild-type human partial length CDKL3 (M1 to D327 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4264220 | B | Binding affinity to wild-type human partial length CDKL3 (M1 to D327 residues) expressed in bacterial expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4307735 | B | Binding affinity to wild-type human partial length CDKL3 (M1 to D327 residues) expressed in bacterial expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4314624 | B | Inhibition of recombinant human full-length CDKL3 (1 to 303 residues) assessed as residual activity at 10 uM using RRRFRPASPLRGP as substrate measured after 120 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4333326 | B | Binding affinity to wild-type human partial length CDKL3 (M1 to D327 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4335016 | B | Inhibition of recombinant full length human CDKL3 assessed as residual activity at 1 uM using RRRFRPASPLRGPPK as substrate incubated for 120 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 19. | ALA4336844 | B | Inhibition of recombinant full length human CDKL3 assessed as residual activity at 10 uM using RRRFRPASPLRGPPK as substrate incubated for 120 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4351797 | B | Inhibition of recombinant human full-length CDKL3 (1 to 303 residues) at 10 uM using RRRFRPASPLRGP as substrate measured after 120 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | single protein format | Scientific Literature |
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