| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1166620 | B | Inhibition of PIK3C2G at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 2. | ALA1175198 | B | Inhibition of PIK3C2G at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 3. | ALA1244566 | B | Binding affinity to PIK3C2G | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 4. | ALA1768740 | B | Binding affinity to PIK3C2G at 1 uM relative to control | 1 | ALA1765054 | single protein format | Scientific Literature | ||
| 5. | ALA1772046 | B | Binding affinity to human PIK3C2G | Homo sapiens | 1 | ALA1770051 | single protein format | Scientific Literature | |
| 6. | ALA1826076 | B | Activity of PIK3C2G kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 7. | ALA1908655 | B | Binding constant for PIK3C2G kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 8. | ALA2154985 | B | Binding affinity to PIK3C2G | 1 | ALA2150858 | single protein format | Scientific Literature | ||
| 9. | ALA2214965 | B | Inhibition of PIK3C2G assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
| 10. | ALA3111951 | B | Inhibition of PIK3C2G (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
| 11. | ALA3119545 | B | Inhibition of PI3KC2gamma (unknown origin) | Homo sapiens | 1 | ALA3112424 | single protein format | Scientific Literature | |
| 12. | ALA3130699 | B | Inhibition of human PI3KC2gamma assessed as residual activity at 1 uM relative to control | Homo sapiens | 3 | ALA3124838 | single protein format | Scientific Literature | |
| 13. | ALA3376671 | B | Inhibition of human PI3KC2gamma by non-radiometric ADP-Glo assay | Homo sapiens | 12 | ALA3352433 | single protein format | Scientific Literature | |
| 14. | ALA3375581 | B | Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity at 10 uM by nonradiometric ADP-Glo assay | Homo sapiens | 41 | ALA3352294 | single protein format | Scientific Literature | |
| 15. | ALA3375584 | B | Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assay | Homo sapiens | 4 | ALA3352294 | single protein format | Scientific Literature | |
| 16. | ALA3789699 | B | Inhibition of N-terminal GST-tagged recombinant human full length PI3KC2gamma expressed in baculovirus infected Sf21 insect cells preincubated for 15 mins followed by addition of cold ATP/gamma32P-ATP measured after 15 mins | Homo sapiens | 2 | ALA3784974 | cell-based format | Scientific Literature | |
| 17. | ALA3861250 | B | Inhibition of PI3KC2gamma (unknown origin) | Homo sapiens | 3 | ALA3860068 | single protein format | Scientific Literature | |
| 18. | ALA3861262 | B | Inhibition of PI3KC2gamma (unknown origin) expressed in HEK293 cells using phosphatidylinositol and gamma-32P-ATP incubated for 20 mins by TLC assay or high-throughput membrane capture assay | Homo sapiens | 4 | ALA3860068 | cell-based format | Scientific Literature | |
| 19. | ALA4025305 | B | Inhibition of wild-type human partial length PIK3C2G (M1 to I1446 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
| 20. | ALA4044116 | B | Inhibition of wild-type human partial length PIK3C2G (M1 to I1446 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature |
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