# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1166053 | B | Inhibition of LZK at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
2. | ALA1174886 | B | Inhibition of LZK at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
3. | ALA1244487 | B | Binding affinity to LZK | 7 | ALA1240346 | single protein format | Scientific Literature | ||
4. | ALA1828395 | B | Activity of LZK kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
5. | ALA1908662 | B | Binding constant for LZK kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
6. | ALA2210638 | B | Inhibition of LZK assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
7. | ALA3111963 | B | Inhibition of LZK (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
8. | ALA4025215 | B | Inhibition of wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
9. | ALA4044026 | B | Inhibition of wild-type human full length LZK (M1 to W966 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
10. | ALA4055105 | B | Inhibition of wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
11. | ALA4119874 | B | Binding affinity to full length wild type human LZK (M1 to W966 residues) expressed in mammalian cells by KINOMEscan assay | Homo sapiens | 2 | ALA4118097 | cell-based format | Scientific Literature | |
12. | ALA4157105 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
13. | ALA4185884 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | cell-based format | Scientific Literature | |
14. | ALA4230784 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
15. | ALA4264373 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature | |
16. | ALA4307883 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4304811 | assay format | Scientific Literature | |
17. | ALA4333470 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4330132 | assay format | Scientific Literature | |
18. | ALA4357962 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4354843 | assay format | Scientific Literature | |
19. | ALA4365800 | B | Inhibition of wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
20. | ALA4382593 | B | Binding affinity to wild-type human full length LZK (M1 to W966 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature |