| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1826633 | B | Activity of MAST1 kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
| 2. | ALA1908788 | B | Binding constant for MAST1 kinase domain | 72 | single protein format | Scientific Literature | |||
| 3. | ALA1166070 | B | Inhibition of MAST1 at 1 uM | 6 | single protein format | Scientific Literature | |||
| 4. | ALA1174903 | B | Inhibition of MAST1 at 10 uM | 2 | single protein format | Scientific Literature | |||
| 5. | ALA1244504 | B | Binding affinity to MAST1 | 7 | single protein format | Scientific Literature | |||
| 6. | ALA2210620 | B | Inhibition of MAST1 assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
| 7. | ALA3111960 | B | Inhibition of MAST1 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4025232 | B | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA4034396 | B | Inhibition of MAST1 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4044043 | B | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA4055217 | B | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 12. | ALA4157122 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA4185901 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 14. | ALA4230801 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4264390 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4307900 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4333487 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4357979 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA4365817 | B | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA4382610 | B | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature |
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