# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1166070 | Binding | Inhibition of MAST1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
2. | ALA1174903 | Binding | Inhibition of MAST1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
3. | ALA1244504 | Binding | Binding affinity to MAST1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
4. | ALA1826633 | Binding | Activity of MAST1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
5. | ALA4357979 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4354843 | assay format | Scientific Literature | |
6. | ALA1908788 | Binding | Binding constant for MAST1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
7. | ALA2210620 | Binding | Inhibition of MAST1 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
8. | ALA3111960 | Binding | Inhibition of MAST1 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
9. | ALA4025232 | Binding | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
10. | ALA4034396 | Binding | Inhibition of MAST1 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
11. | ALA4044043 | Binding | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
12. | ALA4055217 | Binding | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
13. | ALA4157122 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
14. | ALA4185901 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | cell-based format | Scientific Literature | |
15. | ALA4230801 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
16. | ALA4264390 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature | |
17. | ALA4307900 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4304811 | assay format | Scientific Literature | |
18. | ALA4333487 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4330132 | assay format | Scientific Literature | |
19. | ALA4365817 | Binding | Inhibition of wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4364269 | assay format | Scientific Literature | |
20. | ALA4382610 | Binding | Binding affinity to wild-type human partial length MAST1 (S346 to V730 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4382192 | assay format | Scientific Literature |