# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1167697 | B | Inhibition of SBK1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
2. | ALA1175334 | B | Inhibition of SBK1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
3. | ALA1826897 | B | Activity of SBK1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
4. | ALA1908509 | B | Binding constant for SBK1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
5. | ALA2209702 | B | Inhibition of SBK1 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
6. | ALA4025381 | B | Inhibition of wild-type human partial length SBK1 (P23 to P348 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
7. | ALA4044192 | B | Inhibition of wild-type human partial length SBK1 (P23 to P348 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
8. | ALA4055258 | B | Inhibition of wild-type human partial length SBK1 (P23 to P348 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
9. | ALA4157271 | B | Binding affinity to wild-type human partial length SBK1 (P23 to P348 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
10. | ALA4186050 | B | Binding affinity to wild-type human partial length SBK1 (P23 to P348 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | cell-based format | Scientific Literature | |
11. | ALA4230950 | B | Binding affinity to wild-type human partial length SBK1 (P23 to P348 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
12. | ALA4264539 | B | Binding affinity to wild-type human partial length SBK1 (P23 to P348 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature | |
13. | ALA4308048 | B | Binding affinity to wild-type human partial length SBK1 (P23 to P348 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4304811 | assay format | Scientific Literature | |
14. | ALA4314535 | B | Inhibition of recombinant full-length human SBK1 assessed as residual activity at 10 uM using KKLRRTLSVA as substrate measured after 120 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4311992 | single protein format | Scientific Literature | |
15. | ALA4327871 | B | Inhibition of human SBK1 assessed as residual activity at 1 uM using LCGRTGRRNSI as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4325871 | single protein format | Scientific Literature | |
16. | ALA4328235 | B | Inhibition of human SBK1 assessed as residual activity at 100 uM using LCGRTGRRNSI as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
17. | ALA4328599 | B | Inhibition of human SBK1 using LCGRTGRRNSI as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
18. | ALA4333632 | B | Binding affinity to wild-type human partial length SBK1 (P23 to P348 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4330132 | assay format | Scientific Literature | |
19. | ALA4335283 | B | Inhibition of recombinant full-length human SBK1 assessed as residual activity at 1 uM using KKLRRTLSVA as substrate measured after 120 mins in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 2 | ALA4334438 | single protein format | Scientific Literature | |
20. | ALA4337108 | B | Inhibition of recombinant full-length human SBK1 assessed as residual activity at 10 uM using KKLRRTLSVA as substrate incubated for 120 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | ALA4334471 | single protein format | Scientific Literature |