# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1285988 | B | Binding affinity to Influenza A/WSN/33 (H1N1) neuraminidase infected in mouse assessed as half-time for substrate conversion at 10 mg/kg, im administered as single dose | Influenza A virus (A/WSN/1933(H1N1)) | 1 | ALA1275600 | organism-based format | Scientific Literature | |
2. | ALA1285989 | B | Binding affinity to Influenza A/WSN/33 (H1N1) neuraminidase infected in mouse assessed as half-time for substrate conversion at 2 to 20 mg/kg/day, po administered as single dose | Influenza A virus (A/WSN/1933(H1N1)) | 1 | ALA1275600 | organism-based format | Scientific Literature | |
3. | ALA2215924 | B | Inhibition of wild type Influenza A virus A/WSN/1933(H1N1) neuraminidase in virus-infected allantoic fluid using 2'-(4-methylumbelliferyl)-alpha-D-N-acetylneuraminic acid as substrate incubated for 10 mins prior to substrate addition by fluorescence assay | Influenza A virus (A/WSN/1933(H1N1)) | 7 | ALA2203066 | single protein format | Scientific Literature | |
4. | ALA2209787 | B | Inhibition of oseltamivir-resistant Influenza A virus A/WSN/1933/H275Y(H1N1) neuraminidase in virus-infected allantoic fluid using 2'-(4-methylumbelliferyl)-alpha-D-N-acetylneuraminic acid as substrate incubated for 10 mins prior to substrate addition by fluorescence assay | Influenza A virus | 6 | ALA2203066 | single protein format | Scientific Literature | |
5. | ALA2210795 | B | Inhibition of Influenza A virus A/WSN/1933(H1N1)) neuraminidase in the presence of 2'-(4-methyl-umbelliferyl)-alphaD-N-acetylneuraminic acid substrate after 10 mins by fluorometric assay | Influenza A virus (A/WSN/1933(H1N1)) | 17 | ALA2203072 | single protein format | Scientific Literature | |
6. | ALA3267843 | B | Inhibition of neuraminidase H275Y mutant in oseltamivir-resistant Influenza A virus (A/WSN/1933(H1N1)) infected in allantoic fluid of embryonated chicken egg using MUNANA as substrate assessed as release of 4-methylumbelliferone preincubated for 10 mins followed by substrate addition by fluorometric assay | Influenza A virus (A/WSN/1933(H1N1)) | 7 | ALA3259643 | single protein format | Scientific Literature | |
7. | ALA3387279 | B | Inhibition of Influenza A virus A/WSN/1933(H1N1) neuraminidase H275Y mutant using 2-(4-methylumbelliferyl)-alpha-D-N-acetylneuraminic acid after 15 mins by fluorescent assay | Influenza A virus (A/WSN/1933(H1N1)) | 16 | ALA3352719 | single protein format | Scientific Literature | |
8. | ALA3871450 | B | Inhibition of MDCK infected Influenza A virus A/WSN/33(H1N1) neuraminidase using MU-NANA as substrate preincubated for 30 mins followed by substrate addition measured after 1 hr by spectrofluorometric method | Influenza A virus (A/WSN/1933(H1N1)) | 15 | ALA3871267 | cell-based format | Scientific Literature | |
9. | ALA3871451 | B | Competitive inhibition of MDCK infected Influenza A virus A/WSN/33(H1N1) neuraminidase using MU-NANA as substrate preincubated for 30 mins followed by substrate addition measured after 1 hr by spectrofluorometric method | Influenza A virus (A/WSN/1933(H1N1)) | 5 | ALA3871267 | cell-based format | Scientific Literature | |
10. | ALA4155297 | B | Inhibition of Influenza A virus (A/WSN/1933(H1N1)) wild type neuraminidase using MUNANA as substrate preincubated for 10 mins followed by substrate addition and measured for 15 mins by fluorescence assay | Influenza A virus (A/WSN/1933(H1N1)) | 8 | ALA4152278 | single protein format | Scientific Literature | |
11. | ALA4254774 | B | Inhibition of Influenza A virus (A/WSN/1933(H1N1)) neuraminidase pre-incubated for 10 mins before 4-MUNANA substrate addition by fluorometry | Influenza A virus (A/WSN/1933(H1N1)) | 7 | ALA4251642 | single protein format | Scientific Literature | |
12. | ALA4254779 | B | Inhibition of Influenza A virus (A/WSN/1933(H1N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-MUNANA substrate addition by fluorometry | Influenza A virus (A/WSN/1933(H1N1)) | 3 | ALA4251642 | cell-based format | Scientific Literature | |
13. | ALA4262946 | B | Inhibition of Influenza A virus (A/WSN/33(H1N1)) NA up to 100 uM using 4-MUNANA as substrate after 30 mins by fluorescence spectrophotometric assay | Influenza A virus (A/WSN/1933(H1N1)) | 1 | ALA4261546 | single protein format | Scientific Literature |