| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1291121 | B | Displacement of radiolabeled L-[Methyl-14C] from CPT1 at 1 to 3 uM | 1 | ALA1287688 | single protein format | Scientific Literature | ||
| 2. | ALA2216983 | B | Inhibition of CPT1A | 2 | ALA2216752 | single protein format | Scientific Literature | ||
| 3. | ALA2217029 | B | Increase in CPT1A activity in hepatocytes at 60 uM | 1 | ALA2216752 | cell-based format | Scientific Literature | ||
| 4. | ALA2217038 | B | Increase in CPT1 activity in human MCF7 cells assessed as increase in radiolabeled palmitoylcarnitine relative to untreated control | Homo sapiens | 1 | ALA2216752 | cell-based format | Scientific Literature | |
| 5. | ALA2217040 | B | Increase in CPT1 activity in human MCF7 cells assessed as increase in radiolabeled palmitoylcarnitine | Homo sapiens | 1 | ALA2216752 | cell-based format | Scientific Literature | |
| 6. | ALA2217041 | B | Increase in CPT1 activity in human MCF7 cells assessed as increase in radiolabeled palmitoylcarnitine at 31 uM | Homo sapiens | 1 | ALA2216752 | cell-based format | Scientific Literature | |
| 7. | ALA2217044 | B | Increase in muscle CPT1 activity expressed in yeast mitochondrial extracts | 1 | ALA2216752 | tissue-based format | Scientific Literature | ||
| 8. | ALA2217045 | B | Increase in liver CPT1 activity expressed in yeast mitochondrial extracts | 1 | ALA2216752 | tissue-based format | Scientific Literature | ||
| 9. | ALA2217055 | B | Inhibition of CPT1 in liver mitochondria | 1 | ALA2216752 | mitochondrion format | Scientific Literature | ||
| 10. | ALA2217057 | B | Inhibition of CPT1 in heart mitochondria | 1 | ALA2216752 | single protein format | Scientific Literature | ||
| 11. | ALA2217058 | B | Inhibition of human CPT1A expressed in Saccharomyces cerevisiae mitochondria assessed as palmitoylcarnitine by HPLC method | Homo sapiens | 2 | ALA2216752 | mitochondrion format | Scientific Literature | |
| 12. | ALA2217072 | B | Inhibition of human CPT1A | Homo sapiens | 17 | ALA2216752 | single protein format | Scientific Literature | |
| 13. | ALA3431933 | B | SUPPLEMENTARY: Inhibition of Carnitine palmitoyltransferase 1, liver isoform | Homo sapiens | 476 | ALA3431459 | assay format | Deposited Supplementary Bioactivity Data | |
| 14. | ALA4341451 | B | Binding affinity to CPT1A in human A549 cells lysates grown on SILAC media at 10 uM incubated for 1 hr by LC-MS/MS analysis relative to untreated control | Homo sapiens | 1 | ALA4340528 | subcellular format | Scientific Literature |
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