| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3734574 | F | Inhibition of TRPM4 (unknown origin) expressed in HEK293 cells assessed as effect on agonist-induced Ca2+ changes | Homo sapiens | 1 | cell-based format | Patent Bioactivity Data | ||
| 2. | ALA4134892 | B | Inhibition of TRPM4 in human Jurkat T cells assessed as reduction in intracellular calcium flux at 500 nM within 60 mins by whole cell patch clamp electrophysiology method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA4158451 | B | Inhibition of TRPM4 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA4401098 | B | Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dye-based fluorescence assay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 5. | ALA4401099 | B | Inhibition of TRPM4 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA4401100 | B | Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx at 10 uM after 45 mins by ANG2 dye-based fluorescence assay relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA4401101 | B | Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx up to 100 uM after 45 mins by ANG2 dye-based fluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA4411011 | B | Inhibition of TRPM4 channel (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4824111 | B | Agonist activity at human TRPM4 expressed in CHO cells assessed as increase in A23187-induced intracellular calcium level by FLIPR assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 10. | ALA4828444 | B | Antagonist activity at human TRPM4 at <= 30 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA5153236 | B | Agonist activity at human TRPM4 expressed in CHO-K1 cells assessed as increase in relative fluorescence unit by measuring membrane potential by FLIPR assay | Homo sapiens | 9 | cell-based format | Scientific Literature |
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