# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3540644 | ADME | Inhibition of human OATP1B1 expressed HEK293 cells assessed as inhibition of [3H]sulfobromophthalein uptake by liquid scintillation counting | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
2. | ALA3540650 | ADME | Drug uptake in human OATP1B1 expressed HEK293 cells at 20 uM relative to control cells | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
3. | ALA3540652 | ADME | Drug uptake in human OATP1B1 expressed HEK293 cells assessed as net uptake measured per mg of protein | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
4. | ALA3540656 | ADME | Drug uptake in human OATP1B1 expressed HEK293 cells assessed as net uptake | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
5. | ALA3540667 | ADME | Drug uptake in human OATP1B1 expressed HEK293 cells at 20 uM relative to control cells in presence of 100 uM pravastatin | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
6. | ALA3540668 | ADME | Drug uptake in human OATP1B1 expressed HEK293 cells at 20 uM relative to control cells in presence of 10 uM pravastatin | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
7. | ALA3540671 | ADME | Drug uptake in human OATP1B1 expressed HEK293 cells at 20 uM relative to control cells in presence of 100 uM cyclosporine | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
8. | ALA3540674 | ADME | Drug uptake in human OATP1B1 expressed HEK293 cells at 20 uM relative to control cells in presence of 10 to 100 uM budesonide | Homo sapiens | 1 | ALA3525949 | cell-based format | Scientific Literature | |
9. | ALA3537109 | ADME | Inhibition of human OATP1B1 expressed in CHO cells using [3H]estradiol 17beta-D-glucuronide as substrate by liquid scintillation counting analysis | Homo sapiens | 1 | ALA3526034 | cell-based format | Scientific Literature | |
10. | ALA3536606 | ADME | Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction of [3H]E217betaG substrate uptake by liquid scintillation counting | Homo sapiens | 1 | ALA3525903 | cell-based format | Scientific Literature | |
11. | ALA3532587 | ADME | Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction of [3H]estradiol-17beta-glucuronide uptake at 10 uM after 3 mins by beta-counting | Homo sapiens | 6 | ALA3526004 | cell-based format | Scientific Literature | |
12. | ALA3533390 | ADME | Drug uptake in HEK293 cells expressing OATP1B1 (unknown origin) assessed as OATP1B1-mediated drug transport | Homo sapiens | 2 | ALA3525911 | cell-based format | Scientific Literature | |
13. | ALA3533391 | ADME | Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells using pitavastatin substrate | Homo sapiens | 8 | ALA3525911 | cell-based format | Scientific Literature | |
14. | ALA3533735 | ADME | Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells using estradiol-17beta-glucuronide substrate | Homo sapiens | 8 | ALA3525911 | cell-based format | Scientific Literature | |
15. | ALA3533736 | ADME | Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells using estrone-3-sulfate substrate | Homo sapiens | 8 | ALA3525911 | cell-based format | Scientific Literature | |
16. | ALA3533737 | ADME | Drug uptake in HEK293 cells expressing OATP1B1 (unknown origin) assessed as OATP1B1-mediated drug transport per mg protein | Homo sapiens | 2 | ALA3525911 | cell-based format | Scientific Literature | |
17. | ALA3533738 | ADME | Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as protein-mediated pitavastatin uptake | Homo sapiens | 2 | ALA3525911 | cell-based format | Scientific Literature | |
18. | ALA3533751 | ADME | Drug uptake assessed as OATP1B1 (unknown origin)-mediated drug transport expressed in HEK293 cells by LC-MS/MS analysis relative to control | Homo sapiens | 2 | ALA3526031 | cell-based format | Scientific Literature | |
19. | ALA3536013 | ADME | Drug uptake in human OATP1B1 expressing HEK293/PDZK1 cells at 37 degC for 30 mins | Homo sapiens | 1 | ALA3526078 | cell-based format | Scientific Literature | |
20. | ALA3533582 | ADME | Inhibition of OATP1B1-mediated [3H]estrone-3-sulfate uptake in human OATP1B1 expressing HEK293/PDZK1 cells by scintillation counting | Homo sapiens | 2 | ALA3526078 | cell-based format | Scientific Literature |