| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1738450 | U | PUBCHEM_BIOASSAY: Late stage results from the probe development effort to identify inhibitors of the protein methylesterase PME-1: Gel-based Activity-Based Protein Profiling (ABPP) IC50. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2130, AID2143, AID2171, AID2174, AID2177, AID2232, AID2233, AID2291, AID463090, AID463091, AID463124, AID463130, AID463131, AID463132, AID463146, AID463149] Panel member name: APEH Assay Panel member description: Inhibition of N-acylaminoacyl-peptide hydrolase (APEH) (anti-target) | 6 | ALA1201862 | assay format | PubChem BioAssays | ||
| 2. | ALA2027538 | B | Inhibition of APEH in human HeLa cells after 24 hrs | Homo sapiens | 1 | ALA2021843 | cell-based format | Scientific Literature | |
| 3. | ALA2027539 | B | Inhibition of APEH in human A375 cells after 24 hrs | Homo sapiens | 1 | ALA2021843 | cell-based format | Scientific Literature | |
| 4. | ALA2027540 | B | Inhibition of APEH in human HeLa cells at 150 uM after 24 hrs | Homo sapiens | 1 | ALA2021843 | cell-based format | Scientific Literature | |
| 5. | ALA2027541 | B | Inhibition of APEH in human A375 cells at 150 uM after 24 hrs | Homo sapiens | 1 | ALA2021843 | cell-based format | Scientific Literature | |
| 6. | ALA2209095 | B | Inhibition of APEH binding to FP-biotin in [12C][14N]-lysine, arginine and [13C6][15N2]-lysine, arginine labeled HEK293T cells at 20 uM after 1 hr by isotopic activity-based protein profiling-MudPIT assay | Homo sapiens | 1 | ALA2203175 | cell-based format | Scientific Literature | |
| 7. | ALA2212402 | B | Inhibition of acyl peptide hydrolase binding to FP-rhodamine in human HEK293T cells at 0.5 to 50 uM after 30 mins by fluorescence polarization activity-based protein profiling assay | Homo sapiens | 1 | ALA2203175 | cell-based format | Scientific Literature | |
| 8. | ALA4118677 | B | Binding affinity to APEH in human NCI-H23 cells at 1 uM by mass spectrometry based pull down assay | Homo sapiens | 1 | ALA4118021 | cell-based format | Scientific Literature | |
| 9. | ALA4118858 | B | Binding affinity to APEH in human NCI-H358 cells at 1 uM by mass spectrometry based pull down assay | Homo sapiens | 1 | ALA4118021 | cell-based format | Scientific Literature |
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