| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1743314 | A | Major substrate of human cytosolic sulfotransferase SULT1A1 | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 2. | ALA3540601 | A | Activity of human SULT1A1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 3. | ALA3540604 | A | Activity of human SULT1A1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation measured per mg of protein after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA3539752 | A | Drug metabolism assessed as human SULT1A1-mediated (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[1,2-f][1,2,4]triazin-6-yloxy)propane-2-sulfonic acid formation at 2 and 20 uM for 30 mins by LC/MS analysis in presence of PAPS | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA3539757 | A | Activity of human SULT1A1 assessed as compound formation treated with 2 and 20 uM brivanib for 30 mins by LC/MS analysis in presence of PAPS | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA3537867 | A | Activity of human SULT1A1 expressed in Escherichia coli at 20 uM by Michaelis-Menten equation analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA3537868 | A | Activity of human SULT1A1 expressed in Escherichia coli at 20 uM by Michaelis-Menten equation analysis in presence of PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA3537869 | A | Activity of human SULT1A1 expressed in Escherichia coli at 6 uM by Michaelis-Menten equation analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA3537870 | A | Activity of human SULT1A1 expressed in Escherichia coli at 6 uM by Michaelis-Menten equation analysis in presence of PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA3537871 | A | Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescence | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 11. | ALA3537872 | A | Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescence in presence of 3',5'-phosphoadenosine | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 12. | ALA3537873 | A | Inhibition of human SULT1A1 expressed in Escherichia coli assessed as 17beta-estradiol sulfation at 100 nM by Michaelis-Menten equation analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA3537874 | A | Inhibition of human SULT1A1 expressed in Escherichia coli assessed as p-nitrophenol sulfation at 100 nM by Michaelis-Menten equation analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA3537875 | A | Inhibition of human SULT1A1 expressed in Escherichia coli assessed as beta-naphthol sulfation at 100 nM by Michaelis-Menten equation analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA3537876 | A | Inhibition of SULT1A1 in human MCF7 cells assessed as 17beta-estradiol sulfation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA4482682 | B | Inhibition of SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells incubated for 15 mins using para-nitrophenol as substrate by TLC analysis | Homo sapiens | 4 | cell-based format | Patent Bioactivity Data | ||
| 17. | ALA4482692 | B | Substrate activity at SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Km incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | cell-based format | Patent Bioactivity Data | ||
| 18. | ALA4482693 | B | Substrate activity at SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | cell-based format | Patent Bioactivity Data | ||
| 19. | ALA4482694 | B | Substrate activity at SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax/Km ratio incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis | Homo sapiens | 25 | cell-based format | Patent Bioactivity Data |
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