| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA750982 | F | Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4) | 8 | assay format | Scientific Literature | |||
| 2. | ALA750983 | B | KB value was evaluated at the human P2X purinoceptor 4 (P2X4); IA menas inactive | 1 | single protein format | Scientific Literature | |||
| 3. | ALA750984 | F | The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 4 (P2X4) | 1 | assay format | Scientific Literature | |||
| 4. | ALA751124 | F | Inhibition of inward ion current elicited by ATP at human P2X4 receptor (mutant type) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA872178 | F | Inhibitory concentration against human P2X purinoceptor 4 expressed in Xenopus laevis oocytes | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA901769 | B | Activity at human P2X4 receptor at 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 7. | ALA886467 | B | Activity at human P2X4 receptor at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA932850 | B | Inhibition of P2X4 receptor at 10 uM | 1 | single protein format | Scientific Literature | |||
| 9. | ALA982869 | F | Antagonist activity at P2X4 receptor at 10 uM | 1 | assay format | Scientific Literature | |||
| 10. | ALA968798 | B | Activity at P2X4 receptor up to 10 uM | 4 | single protein format | Scientific Literature | |||
| 11. | ALA1017979 | F | Antagonist activity at P2X4 receptor up to 10 uM | 1 | assay format | Scientific Literature | |||
| 12. | ALA960840 | B | Inhibition of P2X4 receptor | 1 | single protein format | Scientific Literature | |||
| 13. | ALA1069596 | F | Antagonist activity at P2X4 receptor | 2 | assay format | Scientific Literature | |||
| 14. | ALA1925629 | B | Inhibition of P2X4 receptor at 10 uM | 1 | single protein format | Scientific Literature | |||
| 15. | ALA2184474 | B | Competitive antagonist activity at human P2X4 receptor expressed in 1321N1 cell membrane assessed as inhibition of [35S]ATPgammaS binding at >10 uM by scintillation counting | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 16. | ALA2184475 | B | Competitive antagonist activity at human P2X4 receptor expressed in 1321N1 cell membrane assessed as inhibition of [35S]ATPgammaS binding by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA2184476 | B | Negative allosteric modulation at human P2X4 receptor expressed in 1321N1 cell membrane assessed as inhibition of [35S]ATPgammaS binding by scintillation counting | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 18. | ALA2184477 | F | Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubated at 100 uM for 30 mins before ATP treatment by Fluo-4 AM fluorescence method | Homo sapiens | 27 | cell-based format | Scientific Literature | ||
| 19. | ALA2184478 | F | Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubated at 10 uM for 30 mins before ATP treatment by Fluo-4 AM fluorescence method | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
| 20. | ALA2184479 | F | Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincubated for 30 mins before ATP treatment by Fluo-4 AM fluorescence method | Homo sapiens | 58 | cell-based format | Scientific Literature |
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