# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1218918 | B | Inhibition of human recombinant matriptase 2 expressed in HEK293 cells in conditioned medium after 20 mins | Homo sapiens | 5 | ALA1212915 | cell-based format | Scientific Literature | |
2. | ALA1218919 | B | Inhibition of human purified matriptase 2 catalytic domain expressed in HEK293 cells after 20 mins | Homo sapiens | 5 | ALA1212915 | cell-based format | Scientific Literature | |
3. | ALA1810434 | B | Inhibition of matriptase 2 | 1 | ALA1806464 | single protein format | Scientific Literature | ||
4. | ALA2090835 | B | Tight binding inhibition of human matriptase2 expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 15 mins prior to substrate addition measured for 30 mins by fluorimetric analysis | Homo sapiens | 1 | ALA2086329 | cell-based format | Scientific Literature | |
5. | ALA2160579 | B | Inhibition of human matriptase-2 expressed in HEK-MT2 cells using fluorogenic Boc- Gln-Ala-Arg-NH-Mec as substrate measured over 400 secs by spectrophotometry | Homo sapiens | 73 | ALA2157883 | cell-based format | Scientific Literature | |
6. | ALA3225092 | B | Inhibition of matriptase-2 (unknown origin) expressed in HEK293 cells using ln-Ala-Arg-a-Arg-para-nitroanilide as substrate by UV-vis spectrophotometry | Homo sapiens | 32 | ALA3217540 | cell-based format | Scientific Literature | |
7. | ALA3371671 | B | Inhibition of human recombinant matriptase-2 using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysis | Homo sapiens | 15 | ALA3351530 | single protein format | Scientific Literature | |
8. | ALA3627229 | B | Inhibition of matriptase (unknown origin) using Ac-RQFRpNA substrate by spectrophotometry method | Homo sapiens | 6 | ALA3621201 | single protein format | Scientific Literature | |
9. | ALA3829337 | B | Inhibition of human matriptase-2 transfected in HEK cells assessed as residual activity at 40 uM using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysis | Homo sapiens | 27 | ALA3826881 | cell-based format | Scientific Literature | |
10. | ALA3829338 | B | Inhibition of human matriptase-2 transfected in HEK cells assessed as residual activity at 5 uM using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysis | Homo sapiens | 1 | ALA3826881 | cell-based format | Scientific Literature | |
11. | ALA3829805 | B | Inhibition of human matriptase-2 transfected in HEK cells using Boc-Gln-Ala-Arg-AMC as substrate after 20 mins by fluorimetric analysis | Homo sapiens | 7 | ALA3826881 | cell-based format | Scientific Literature | |
12. | ALA4009363 | B | Inhibition of recombinant human C-terminal V5-His-tagged matriptase-2 expressed in Drosophila S2 cells using Boc-Gln-Ala-ArgAMC as substrate measured for 1200 mins by fluorescence assay | Homo sapiens | 29 | ALA4007428 | cell-based format | Scientific Literature | |
13. | ALA4009366 | B | Reversible inhibition of recombinant human C-terminal V5-His-tagged matriptase-2 expressed in Drosophila S2 cells assessed as dissociation half time using Boc-Gln-Ala-ArgAMC as substrate measured for 1200 mins by fluorescence assay | Homo sapiens | 3 | ALA4007428 | cell-based format | Scientific Literature | |
14. | ALA5256566 | B | Inhibition of recombinant human matriptase 2 using Boc-Gln-Ala-Arg-AMC as substrate at 3.85 to 385 nM preincubated for 30 mins followed by substrate addition and measured for 40 mins by microplate reader method | Homo sapiens | 4 | ALA5252656 | single protein format | Scientific Literature |