| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1832846 | B | Binding affinity to PB1 assessed as change in melting temperature at 100 uM by differential scanning fluorimetry | 9 | ALA1828554 | single protein format | Scientific Literature | ||
| 2. | ALA1958935 | B | Binding affinity to PB1 assessed as change in melting temperature at 100 uM by protein stability shift assay | 12 | ALA1955750 | single protein format | Scientific Literature | ||
| 3. | ALA1958944 | B | Binding affinity to PB1 assessed as change in melting temperature at 10 uM by protein stability shift assay | 6 | ALA1955750 | single protein format | Scientific Literature | ||
| 4. | ALA2183671 | B | Binding affinity to pb1 isoform 5 assessed as change in melting temperature at 10 uM by thermal shift assay | 1 | ALA2177039 | single protein format | Scientific Literature | ||
| 5. | ALA3111328 | B | Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) at 100 uM by AlphaScreen assay relative to control | Homo sapiens | 4 | ALA3108763 | single protein format | Scientific Literature | |
| 6. | ALA3111331 | B | Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assay | Homo sapiens | 4 | ALA3108763 | single protein format | Scientific Literature | |
| 7. | ALA3111338 | B | Binding affinity to PB1-5 bromodomain (unknown origin) assessed as change in melting temperature at 10 uM by differential scanning fluorimetric analysis | Homo sapiens | 35 | ALA3108763 | single protein format | Scientific Literature | |
| 8. | ALA3226592 | B | Binding affinity to PB1-5 bromodomain (unknown origin) assessed as change in melting temperature at 10 uM by differential scanning fluorimetric analysis | Homo sapiens | 1 | ALA3217564 | single protein format | Scientific Literature | |
| 9. | ALA3383426 | B | Inhibition of human PBRM1 bromodomain 1 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
| 10. | ALA3383427 | B | Inhibition of human PBRM1 bromodomain 5 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
| 11. | ALA3583525 | B | Binding affinity to biotinylated PB1BR5 (645 to 766 amino acid residues) (unknown origin) expressed in Rosetta2 cells by bio-layer interferometry method | Homo sapiens | 1 | ALA3580597 | cell-based format | Scientific Literature | |
| 12. | ALA3591399 | B | Binding affinity to PBRM1 in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 3 | ALA3588744 | cell-based format | Scientific Literature | |
| 13. | ALA3757231 | B | Inhibition of PB1 bromodomain-5 (unknown origin) by isothermal titration calorimetry | Homo sapiens | 1 | ALA3751772 | single protein format | Scientific Literature | |
| 14. | ALA3773272 | B | Binding affinity to biotinylated PB1 bromodomain-1 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 15. | ALA3773273 | B | Binding affinity to biotinylated PB1 bromodomain-2 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 16. | ALA3773274 | B | Binding affinity to biotinylated PB1 bromodomain-4 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 17. | ALA3773275 | B | Binding affinity to biotinylated PB1 bromodomain-5 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 18. | ALA3773276 | B | Binding affinity to biotinylated PB1 bromodomain-6 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 19. | ALA3777037 | B | Inhibition of recombinant human PBRM1 bromodomain 2 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 20. | ALA3777038 | B | Inhibition of recombinant human PBRM1 bromodomain 5 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature |
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