# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1832849 | B | Binding affinity to BRDT assessed as change in melting temperature at 100 uM by differential scanning fluorimetry | 9 | single protein format | Scientific Literature | |||
2. | ALA1958931 | B | Binding affinity to BRDT-BD1 assessed as change in melting temperature at 100 uM by protein stability shift assay | 12 | single protein format | Scientific Literature | |||
3. | ALA1958940 | B | Binding affinity to BRDT-BD1 assessed as change in melting temperature at 10 uM by protein stability shift assay | 6 | single protein format | Scientific Literature | |||
4. | ALA1958563 | B | Binding affinity to BRDT-BD1 by isothermal titration calorimetry | 1 | single protein format | Scientific Literature | |||
5. | ALA2183672 | B | Binding affinity to BRDT isoform 1 assessed as change in melting temperature at 10 uM by thermal shift assay | 1 | single protein format | Scientific Literature | |||
6. | ALA3383418 | B | Inhibition of human BRDT bromodomain 1 by BROMOscan assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
7. | ALA3383419 | B | Inhibition of human BRDT bromodomain 2 by BROMOscan assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA3384679 | B | Inhibition of BRDT (unknown origin) by TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
9. | ALA3587530 | B | Binding affinity to 6-His-FLAG-Tev-BRDT BD1 (1 to 397) (unknown origin) harboring BD2 Y309A mutant | Homo sapiens | 2 | single protein format | Scientific Literature | ||
10. | ALA3587531 | B | Binding affinity to 6-His-FLAG-Tev-BRDT BD2 (1 to 397) (unknown origin) harboring BD1 Y66A mutant | Homo sapiens | 2 | single protein format | Scientific Literature | ||
11. | ALA3591395 | B | Binding affinity to BRDT in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
12. | ALA3591405 | B | Binding affinity to BRDt containing BD1 bromodomains (unknown origin) by TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
13. | ALA3592018 | B | Binding affinity to BRDt containing BD2 bromodomains (unknown origin) by TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
14. | ALA3773118 | B | Binding affinity to biotinylated BRDT bromodomain-1 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | assay format | Scientific Literature | ||
15. | ALA3773119 | B | Binding affinity to biotinylated BRDT bromodomain-2 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | assay format | Scientific Literature | ||
16. | ALA3777030 | B | Inhibition of recombinant human BRDT bromodomain 1 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
17. | ALA3777031 | B | Inhibition of recombinant human BRDT bromodomain 2 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
18. | ALA3778792 | B | Inhibition of GST-tagged human BRDT bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
19. | ALA3782666 | B | Binding affinity to human His6-tagged BRDT bromodomain 1 (N21 to E137 residues) expressed in Escherichia coli BL21(DE3) cells at 200 uM incubated for 30 mins by SYPRO orange staining based fluorescence thermal shift assay | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
20. | ALA3825273 | B | Activity at human BRD-T up to 100 uM by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature |