| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1174099 | B | Inhibition of CASK at 10 uM | 2 | single protein format | Scientific Literature | |||
| 2. | ALA1908446 | B | Binding constant for CASK kinase domain | 72 | single protein format | Scientific Literature | |||
| 3. | ALA2209342 | B | Inhibition of CASK assessed as residual activity at 10 uM relative to control | 1 | single protein format | Scientific Literature | |||
| 4. | ALA2422451 | B | Inhibition of CASK in human PC3 cell lysates at 10 uM using desthiobiotin-tagged ATP probe AX9989 followed by trypsinization by LC/MS analysis | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 5. | ALA4025046 | B | Inhibition of wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA4034281 | B | Inhibition of CASK Lysine 1 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA4043857 | B | Inhibition of wild-type human partial length CASK (M1 to H315 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA4055131 | B | Inhibition of wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 9. | ALA4118316 | B | Inhibition of CASK in human SKCO1 cells at 1 uM after 4 hrs using biotin labeled ETGQQFAVKIVDVAK probe by mass-spectrometric analysis relative to control | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 10. | ALA4156936 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA4185715 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 12. | ALA4230615 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA4264204 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4307720 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4322759 | B | Binding affinity to recombinant N-terminal His-FLAG-GST-tagged CASK (unknown origin) (1 to 570 residues) expressed in baculovirus infected Sf9 insect cells incubated for 1 hr by TR-FRET assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 16. | ALA4333311 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4357793 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4365638 | B | Inhibition of wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA4382424 | B | Binding affinity to wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA4389143 | B | Inhibition of wild-type human partial length CASK (M1 to H315 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature |
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