# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1166832 | B | Inhibition of PRP4 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
2. | ALA1175242 | B | Inhibition of PRP4 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
3. | ALA1244947 | B | Binding affinity to PRP4 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
4. | ALA1826693 | B | Activity of PRP4 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
5. | ALA1908447 | B | Binding constant for PRP4 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
6. | ALA2212021 | B | Inhibition of PRP4 assessed as residual activity at 10 uM relative to control | 1 | ALA2203081 | single protein format | Scientific Literature | ||
7. | ALA2424233 | B | Inhibition of PRP4 in human PC3 cell lysates at 10 uM using desthiobiotin-tagged ATP probe AX9989 followed by trypsinization by LC/MS analysis | Homo sapiens | 12 | ALA2417377 | single protein format | Scientific Literature | |
8. | ALA3111940 | B | Inhibition of PRP4 (unknown origin) assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3108735 | single protein format | Scientific Literature | |
9. | ALA4025350 | B | Inhibition of wild-type human partial length PRP4 (D657 to I1007 residues) expressed in bacterial expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
10. | ALA4034474 | B | Inhibition of PRP4 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
11. | ALA4034543 | B | Inhibition of PRP4 (unknown origin) labeling at protein kinase domain at 10 uM relative to control | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
12. | ALA4044161 | B | Inhibition of wild-type human partial length PRP4 (D657 to I1007 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | assay format | Scientific Literature | |
13. | ALA4045813 | B | Inhibition of PRP4 (AAGIGKDFKENPNLR) in human PBMC at 1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
14. | ALA4046054 | B | Inhibition of PRP4 (AAGIGKDFKENPNLR) in human PBMC at 0.1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
15. | ALA4055118 | B | Inhibition of wild-type human partial length PRP4 (D657 to I1007 residues) expressed in bacterial expression system assessed as residual activity at 50 nM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4052645 | assay format | Scientific Literature | |
16. | ALA4118460 | B | Inhibition of PRP4 in human SKCO1 cells at 1 uM after 4 hrs using biotin labeled CNILHADIKPDNILVNESK probe by mass-spectrometric analysis relative to control | Homo sapiens | 3 | ALA4118021 | cell-based format | Scientific Literature | |
17. | ALA4157240 | B | Binding affinity to wild-type human partial length PRP4 (D657 to I1007 residues) expressed in bacterial expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
18. | ALA4186019 | B | Binding affinity to wild-type human partial length PRP4 (D657 to I1007 residues) expressed in Escherichia coli BL21 at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | assay format | Scientific Literature | |
19. | ALA4191160 | B | Inhibition of recombinant human PRP4 (663 to end residues) at 1 uM using casein as substrate after 120 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4190187 | single protein format | Scientific Literature | |
20. | ALA4230919 | B | Binding affinity to wild-type human partial length PRP4 (D657 to I1007 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature |