| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1175191 | B | Inhibition of Plasmodium falciparum PFCDPK1 at 10 uM | Plasmodium falciparum | 2 | single protein format | Scientific Literature | ||
| 2. | ALA1908456 | B | Binding constant for PFCDPK1(P.falciparum) kinase domain | 72 | single protein format | Scientific Literature | |||
| 3. | ALA2215407 | B | Inhibition of Plasmodium falciparum PFCDPK1 assessed as residual activity at 10 uM relative to control | Plasmodium falciparum | 1 | single protein format | Scientific Literature | ||
| 4. | ALA3301566 | F | MMV: CDPK1 Protein kinase inhibition assay using recombinant PfCDPK1, syntide 2 peptide substrate, ATP and KinaseGlo to measure % inhibition at 1 uM MMV box compound. | Plasmodium falciparum | 400 | assay format | MMV Malaria Box | ||
| 5. | ALA3562142 | F | PubChem BioAssay. Biochemical screen of P. falciparum CDPK1. (Class of assay: confirmatory) | 181 | assay format | PubChem BioAssays | |||
| 6. | ALA4025298 | B | Inhibition of wild-type Plasmodium falciparum isolate 3D7 full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 7. | ALA4149569 | B | Inhibition of Plasmodium falciparum recombinant CDPK1 expressed in Escherichia coli expression system after 1 hr in presence of [gamma33P]ATP by scintillation proximity assay | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 8. | ALA4149571 | B | Inhibition of Plasmodium falciparum recombinant His-tagged CDPK1 expressed in Escherichia coli BL21(DE3) after 1 hr in presence of [gamma33P]ATP by scintillation proximity assay | Plasmodium falciparum | 2 | assay format | Scientific Literature | ||
| 9. | ALA4157188 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 10. | ALA4185967 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 2 | cell-based format | Scientific Literature | ||
| 11. | ALA4230867 | B | Binding affinity to wild-type Plasmodium falciparum 3D7 full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum 3D7 | 1 | assay format | Scientific Literature | ||
| 12. | ALA4264456 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 13. | ALA4307966 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 14. | ALA4333551 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 15. | ALA4358045 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 16. | ALA4365883 | B | Inhibition of wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 17. | ALA4382676 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 18. | ALA4389395 | B | Inhibition of wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 19. | ALA4389872 | B | Inhibition of wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
| 20. | ALA4391498 | B | Binding affinity to wild-type Plasmodium falciparum full length CDPK1 (M1 to S524 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature |
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