# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1908457 | B | Binding constant for PFPK5(P.falciparum) kinase domain | 72 | single protein format | Scientific Literature | |||
2. | ALA4025299 | B | Inhibition of wild-type Plasmodium falciparum isolate 3D7 full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
3. | ALA4157189 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
4. | ALA4185968 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 2 | cell-based format | Scientific Literature | ||
5. | ALA4230868 | B | Binding affinity to wild-type Plasmodium falciparum 3D7 full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum 3D7 | 1 | assay format | Scientific Literature | ||
6. | ALA4264457 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
7. | ALA4307967 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
8. | ALA4333552 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
9. | ALA4358046 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
10. | ALA4365884 | B | Inhibition of wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
11. | ALA4382677 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
12. | ALA4389396 | B | Inhibition of wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
13. | ALA4389873 | B | Inhibition of wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system at 1 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
14. | ALA4391499 | B | Binding affinity to wild-type Plasmodium falciparum full length PK5 (M1 to N288 residues) expressed in mammalian expression system assessed as residual binding level at 10 uM by Kinomescan method relative to control | Plasmodium falciparum | 1 | assay format | Scientific Literature | ||
15. | ALA4879872 | B | KinomeScan assay: inhibition of PFPK5(P.falciparum) | Plasmodium falciparum | 108 | single protein format | Donated Chemical Probes - SGC Frankfurt |