| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1912611 | B | Irreversible inhibition of PAD1 assessed as citrulline formation at 1 mM measured after 20 hrs by colorimetric assay in presence of 2 mM benzoyl-L-arginine ethyl ester | 2 | single protein format | Scientific Literature | |||
| 2. | ALA1913984 | B | Irreversible inhibition of PAD1 assessed as citrulline formation at 1 mM measured after 20 hrs by colorimetric assay in presence of 10 mM benzoyl-L-arginine ethyl ester | 2 | single protein format | Scientific Literature | |||
| 3. | ALA1914035 | B | Ratio of Kinact to Ki for F-amidine to compound for PAD1 | 1 | single protein format | Scientific Literature | |||
| 4. | ALA1914039 | B | Ratio of Kinact to Ki for Cl-amidine to compound for PAD1 | 1 | single protein format | Scientific Literature | |||
| 5. | ALA1914012 | B | Irreversible inhibition of PAD1 assessed as hydrolysis of benzoyl-L-arginine ethyl ester preincubated for 15 mins measured after 15 mins by fluorometric analysis | 4 | single protein format | Scientific Literature | |||
| 6. | ALA1914015 | B | Irreversible inhibition of PAD1 assessed as residual activity at 1 mM measured after 20 hrs by colorimetric assay | 4 | single protein format | Scientific Literature | |||
| 7. | ALA1914105 | B | Irreversible inhibition of PAD1 assessed as residual activity measured after 20 hrs by colorimetric assay | 3 | single protein format | Scientific Literature | |||
| 8. | ALA1914109 | B | Ratio of Kinact to Ki for PAD1 | 4 | single protein format | Scientific Literature | |||
| 9. | ALA2212449 | B | Irreversible inhibition of PAD1 for 1 hr by dialysis | 2 | single protein format | Scientific Literature | |||
| 10. | ALA2212450 | B | Irreversible inhibition of PAD1 at 15 to 500 uM after 30 mins by competitive ABPP assay | 2 | single protein format | Scientific Literature | |||
| 11. | ALA2212942 | B | Ratio of Kinact to Ki for PAD1 | 11 | single protein format | Scientific Literature | |||
| 12. | ALA2328663 | B | Ratio of Kinact to Ki for human PAD1 using BAEE as substrate after 30 mins | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 13. | ALA3117926 | B | Ratio of Kinact to Ki(app) for recombinant wild-type PAD1 (unknown origin) using N-alpha-Benzoyl-L-arginine amide as substrate preincubated for 10 mins followed by substrate addition measured after 15 mins by COLDER assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 14. | ALA3119090 | B | Irreversible inhibition of recombinant wild-type PAD1 (unknown origin) using N-alpha-Benzoyl-L-arginine amide as substrate assessed as residual activity at 170-fold excess of compound after 1 hr by dialysis method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3119095 | B | Inhibition of recombinant wild-type PAD1 (unknown origin) using N-alpha-Benzoyl-L-arginine amide as substrate preincubated for 15 mins followed by substrate addition measured after 15 mins by COLDER assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 16. | ALA3119099 | B | Inhibition of recombinant wild-type PAD1 (unknown origin) using N-alpha-Benzoyl-L-arginine amide as substrate assessed as residual activity at 10 uM preincubated for 15 mins followed by substrate addition measured after 15 mins by COLDER assay relative to control | Homo sapiens | 32 | single protein format | Scientific Literature | ||
| 17. | ALA3413585 | B | Ratio of Kinact to Ki for PAD1 (unknown origin) using N-alpha-benzoyl-L-arginine ethyl ester as substrate assessed as citrulline production after 15 mins by COLDER assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA3414097 | B | Inhibition of PAD1 (unknown origin) using N-alpha-benzoyl-L-arginine ethyl ester as substrate assessed as citrulline production after 15 mins by COLDER assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA4026701 | B | Inhibition of full length human GST-tagged PAD1 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate addition measured after 30 mins | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 20. | ALA4029649 | B | Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assay | Homo sapiens | 4 | single protein format | Scientific Literature |
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