| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1942534 | B | Inhibition of KDM3A | 1 | single protein format | Scientific Literature | |||
| 2. | ALA3110469 | B | Inhibition of recombinant JMJD1A (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen method | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 3. | ALA3591678 | B | Inhibition of JMJD1A (unknown origin) using H3K9mel peptide | Homo sapiens | 17 | single protein format | Scientific Literature | ||
| 4. | ALA3624700 | B | Inhibition of KDM3A (unknown origin) using H3(1-21)K9Me2-GGK-biotin substrate incubated for 5 mins by alpha screen assay | Homo sapiens | 32 | single protein format | Scientific Literature | ||
| 5. | ALA3624710 | B | Inhibition of KDM3A (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 6. | ALA3776337 | B | Inhibition of KDM3A (unknown origin) expressed in Escherichia coli using H3 (1 to 21 residues) K9Me2-GGK-Biotin KDM3A Cognate Ligand/10 uM alpha-ketoglutarate as substrate/cofactor preincubated for 5 mins followed by substrate addition measured after 20 mins by alphascreen assay | Homo sapiens | 6 | assay format | Scientific Literature | ||
| 7. | ALA3776390 | B | Inhibition of KDM3A (unknown origin) using biotin-H3K9me2 (1 to 21 residues) as substrate preincubated for 15 mins followed by substrate addition measured after 5 mins by alphascreen assay | Homo sapiens | 7 | single protein format | Scientific Literature | ||
| 8. | ALA3791193 | B | Inhibition of KDM3A (unknown origin) after 24 hrs by alphascreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA3791434 | B | Inhibition of KDM3A (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA3789207 | B | Inhibition of recombinant human N-terminal FLAG-tagged KDM3A (2 to 1322 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me as substrate preincubated for 10 mins followed by substrate addition measured after 10 mins by AlphaLisa assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 11. | ALA3795793 | B | Inhibition of KDM3A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of substrate peptide/ ascorbate/2-OG/ Fe(2) measured after 1 hr by AlphaLISA method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA3859078 | B | Inhibition of KDM3A (unknown origin) at 10 uM using biotin-labeled H3K4me1 (1 to 21) peptide and SAM as substrate measured after 30 mins by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4193851 | B | Inhibition of KDM3A (unknown origin) using biotinylated H3K9me1 peptide and alpha-ketoglutarate as substrate measured after 20 mins by LANCE TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA4195559 | B | Inhibition of recombinant human C-terminal FLAG-tagged JMJD1A (2 to 1321 residues) expressed in baculovirus infected Sf9 cells at 10 uM relative to control | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 15. | ALA4223298 | B | Inhibition of KDM3A (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4316553 | B | Inhibition of Flag-tagged KDM3A (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as formaldehyde release using core histone as substrate preincubated with enzyme for 10 mins followed by incubation with substrate for 1 hr measured following 2 hrs incubation with ammonium acetate/acetoacetanilide by fluorescence based analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4353693 | B | Inhibition of KDM3A (unknown origin) by Alphascreen assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 18. | ALA4424788 | B | Inhibition of human N-terminal FLAG-tagged KDM3A (2 to 1321 residues) expressed in baculovirus infected Sf9 insect cells at 50 uM using H3(1-21)K9(Me1)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 19. | ALA4424789 | B | Inhibition of human N-terminal FLAG-tagged KDM3A (2 to 1321 residues) expressed in baculovirus infected Sf9 insect cells at 25 uM using H3(1-21)K9(Me1)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 20. | ALA4424797 | B | Inhibition of human N-terminal FLAG-tagged KDM3A (2 to 1321 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K9(Me1)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay | Homo sapiens | 1 | cell-based format | Scientific Literature |
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