| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1942536 | B | Inhibition of KDM2A | 2 | single protein format | Scientific Literature | |||
| 2. | ALA2167327 | B | Mixed type inhibition of human KDM2A expressed in Escherichia coli assessed inhibition constant for compound-enzyme-substrate complex using methyl lysine peptide substrate by enzyme kinetic assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 3. | ALA2167328 | B | Competitive inhibition of human KDM2A expressed in Escherichia coli using 2-oxoglutarate by enzyme kinetic assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA2167513 | B | Inhibition of human KDM2A expressed in Escherichia coli by formaldehyde dehydrogenase coupled assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA2167522 | B | Inhibition of human KDM2A expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assay | Homo sapiens | 10 | assay format | Scientific Literature | ||
| 6. | ALA2318587 | B | Displacement of 2OG from FBXL11 (1 to 517) (unknown origin) expressed in Escherichia coli at 800 uM | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 7. | ALA2395580 | B | Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to compound addition measured after 4 hrs by fluorescence polarization assay in presence of H3K36me2 peptide | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA2395581 | B | Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to compound addition measured after 4 hrs by fluorescence polarization assay in presence of N-oxalyl glycine | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA2395582 | B | Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to compound addition measured after 4 hrs by fluorescence polarization assay in presence of pyridine 2,4-dicarboxylic acid | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA2395583 | B | Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to compound addition measured after 4 hrs by fluorescence polarization assay in presence of alpha-ketoglutarate | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA2395584 | B | Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 after 4 to 24 hrs by fluorescence polarization assay in presence of Ni2+ | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA2396328 | B | Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assay in presence of Co2+ | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA2396329 | B | Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assay in presence of Ni2+ | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA2396330 | B | Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA2396331 | B | Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 under anaerobic conditions by fluorescence polarization assay in presence of Fe2+ | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA2396334 | B | Inhibition of recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 using SAPATGGVK(Me2)KPHRYRPGTVAL as substrate incubated for 15 mins prior to substrate addition measured after 50 mins by rapid fire mass spectrophotometric analysis | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 17. | ALA2396335 | B | Competitive binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 incubated for 30 mins prior to compound addition measured after 4 hrs by fluorescence polarization assay in presence of methylstat acid | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA2396336 | B | Binding affinity to recombinant 6xHis-tagged JHDM1A (unknown origin) expressed in Escherichia coli BL21 by fluorescence polarization assay in presence of Fe2+ and sodium ascorbate | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA2427605 | B | Inhibition of KDM2A (unknown origin) | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 20. | ALA5141184 | B | Inhibition of KDM2A in human MIA PaCa-2 cells assessed as induction of H3K36me2 measured by immunofluorescence assay | Homo sapiens | 3 | cell-based format | Scientific Literature |
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