# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1942759 | B | Inhibition of human PRPK in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM | Homo sapiens | 4 | ALA1938230 | cell-based format | Scientific Literature | |
2. | ALA2424037 | B | Inhibition of PRPK in human PC3 cell lysates at 10 uM using desthiobiotin-tagged ATP probe AX9989 followed by trypsinization by LC/MS analysis | Homo sapiens | 12 | ALA2417377 | single protein format | Scientific Literature | |
3. | ALA3991917 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 243 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
4. | ALA4034475 | B | Inhibition of PRPK ATP binding site (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4033637 | single protein format | Scientific Literature | |
5. | ALA4045814 | B | Inhibition of PRPK ATP binding site (FLSGLELVKQGAEAR) in human PBMC at 1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
6. | ALA4046055 | B | Inhibition of PRPK ATP binding site (FLSGLELVKQGAEAR) in human PBMC at 0.1 uM | Homo sapiens | 1 | ALA4043168 | single protein format | Scientific Literature | |
7. | ALA4118461 | B | Inhibition of PRPK in human SKCO1 cells at 1 uM after 4 hrs using biotin labeled FLSGLELVKQGAEAR probe by mass-spectrometric analysis relative to control | Homo sapiens | 3 | ALA4118021 | cell-based format | Scientific Literature | |
8. | ALA4804481 | B | Inhibition of PRPK in human NCI-H929 cells by mass spectroscopic analysis | Homo sapiens | 6 | ALA4804281 | cell-based format | Patent Bioactivity Data | |
9. | ALA4804663 | B | Inhibition of PRPK in human NCI-H929 cells at 10 uM by mass spectroscopic analysis relative to control | Homo sapiens | 6 | ALA4804281 | cell-based format | Patent Bioactivity Data |