# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1948736 | B | Binding affinity to LMPX/beta2 in mouse EL4 cells at 10 uM after 1.5 hrs by Western blotting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
2. | ALA3864641 | B | Inhibition of chymotrypsin-like activity of 20S proteasome in mouse blood at 0.5 to 12.5 uM preincubated for 40 mins followed by addition of Suc-Leu-Leu-Val-Tyr-AMC as substrate relative to control | Mus musculus | 5 | tissue-based format | Scientific Literature | ||
3. | ALA4003670 | B | Inhibition of chymotrypsin-like activity of 20S proteasome in mouse blood at 0.5 uM pretreated for 40 mins followed by Suc-Leu-Leu-Val-Tyr-AMC substrate addition by fluorescence assay | Mus musculus | 4 | single protein format | Scientific Literature | ||
4. | ALA4003675 | B | Inhibition of chymotrypsin-like activity of 20S proteasome in mouse blood at 2.5 uM pretreated for 40 mins followed by Suc-Leu-Leu-Val-Tyr-AMC substrate addition by fluorescence assay relative to control | Mus musculus | 7 | single protein format | Scientific Literature | ||
5. | ALA4411754 | B | Inhibition of 20S proteosome beta 5 in mouse A20 cells by ELISA | Mus musculus | 12 | cell-based format | Scientific Literature |