| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2061147 | B | Binding affinity to FKBP51 FK1 domain by competitive fluorescence polarization assay | Homo sapiens | 42 | single protein format | Scientific Literature | ||
| 2. | ALA2061150 | B | Binding affinity to FKBP51 FK1 domain by fluorescence polarization assay | Homo sapiens | 28 | single protein format | Scientific Literature | ||
| 3. | ALA5253378 | B | Binding affinity to FKBP51 (unknown origin) | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 4. | ALA5253391 | B | Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 5. | ALA2351896 | B | Binding affinity to human His-tagged FKBP51 FK1 domain (1 to 140) by isothermal titration calorimetric analysis | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA2351897 | B | Binding affinity to FKBP51 (unknown origin) assessed as increase in [3H]-dexamethasone binding to glucocorticoid receptor | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 7. | ALA2351899 | B | Binding affinity to human FKBP51 by competitive fluorescence polarization assay | Homo sapiens | 27 | single protein format | Scientific Literature | ||
| 8. | ALA3624906 | B | Binding affinity to FKBP51 (unknown origin) by competitive fluorescence polarization assay | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 9. | ALA3624909 | B | Displacement of iFit-FL from FKBP51 (unknown origin) by fluorescence polarization assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 10. | ALA3795199 | B | Binding affinity to FKBP51 FK506-binding domain (1 to 140 amino acids) (unknown origin) incubated for 30 mins using fluorescein-conjugated 2-(5-((2-(3-((R)-3-(3,4-dimethoxyphenyl)-1-((S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carbonyloxy)propyl)phenoxy)acetamido)methyl)-6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid by competitive fluorescence polarization assay | Homo sapiens | 39 | single protein format | Scientific Literature | ||
| 11. | ALA3795202 | B | Binding affinity to FKBP51 (unknown origin) by competitive fluorescence polarization assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 12. | ALA4048818 | B | Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)propylcarbamoyl)-2-(6-(dimethylamino)-3-(dimethyliminio)-3,10-dihydroanthracen-9-yl)benzoate from human FKBP51 after 30 mins by fluorescence polarization assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4379896 | B | Inhibition of human full length N-terminal His-tagged/C-terminal FLAG tagged FKBP51 expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by competitive fluorescence polarization assay | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
| 14. | ALA4379919 | B | Inhibition of human full length N-terminal His-tagged/C-terminal FLAG tagged FKBP51 expressed in Escherichia coli BL21 (DE3) cells at >=10 uM incubated for 30 mins by competitive fluorescence polarization assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 15. | ALA4606613 | B | Binding affinity to 15N-labeled FKBP51 (1 to 140 residues) (unknown origin) expressed in Escherichia coli OD2N assessed as induction of chemical shift perturbations by two-dimensional 1H/15N HSQC NMR spectroscopy | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 16. | ALA4606614 | B | Binding affinity to 15N-labeled FKBP51 (1 to 140 residues) (unknown origin) expressed in Escherichia coli OD2N assessed as induction of chemical shift perturbations at Ile87 residues by two-dimensional 1H/15N HSQC NMR spectroscopy | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 17. | ALA4606615 | B | Binding affinity to 15N-labeled FKBP51 (1 to 140 residues) (unknown origin) expressed in Escherichia coli OD2N assessed as induction of chemical shift perturbations at Leu81, Gly82, Gln85, Ile87, Ala89, Trp90, Asp91, Met97, and Glu110 residues by two-dimensional 1H/15N HSQC NMR spectroscopy | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4606616 | B | Binding affinity to 15N-labeled FKBP51 (1 to 140 residues) (unknown origin) expressed in Escherichia coli OD2N by two-dimensional 1H/15N HSQC NMR spectroscopy | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 19. | ALA4835123 | B | Displacement of fluorescent tracer 5-(3-(4-((1S,5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-3-(pyridin-3-ylmethyl)-3,10-diazabicyclo[4.3.1]decan-5-yl)-1H-1,2,3-triazol-1-yl)propylcarbamoyl)-2-(6-(dimethylamino)-3-(dimethyliminio)-3H-xanthen-9-yl)benzoate from recombinant full length C-terminal FLAG-tagged FKBP51 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by fluorescence polarisation competition binding assay | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
| 20. | ALA4835130 | B | Binding affinity to FKBP51 FK1 domain (unknown origin) assessed as dissociation constant at 25 degreeC by isothermal titration calorimetric analysis | Homo sapiens | 2 | single protein format | Scientific Literature |
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