| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2071961 | B | Inhibition of KDM6A | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA2427606 | B | Inhibition of human recombinant KDM6A after 1 hr | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 3. | ALA3782534 | B | Inhibition of human KDM6A preincubated for 10 mins followed by substrate addition by AlphaLISA assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 4. | ALA3789214 | B | Inhibition of KDM6A (919 to 1401 residues) (unknown origin) expressed in Escherichia coli using biotinylated histone H3 as substrate preincubated for 10 mins followed by substrate addition measured after 10 mins by AlphaLisa assay | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 5. | ALA4035841 | B | Inhibition of recombinant human N-terminal FLAG-tagged KDM6A expressed in baculovirus infected Sf9 insect cells using H3K27me3 peptide as substrate after 30 to 45 mins by TR-FRET assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 6. | ALA4270047 | B | Inhibition of KDM6A (880 to 1401 residues) (unknown origin) using H3 ( 21 to 44 residues) K27me3 as substrate preincubated for 15 min followed by substrate addition measured after 15 mins by FDH-coupled demethylase assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 7. | ALA4427168 | B | Inhibition of KDM6A (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4433873 | B | Inhibition of UTX (unknown origin) using histone H3 peptide as substrate incubated for 30 mins followed by substrate addition by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4832327 | B | Inhibition of KDM6A (unknown origin) by AlphaLISA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA5127962 | B | Inhibition of KDM6A (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA5210083 | F | Affinity Phenotypic Cellular interaction (Inhibition of TNF release (in LPS stimulated human macrophages derived from PBMC)) EUB0000217b KDM6A/UTX | Homo sapiens | 1 | assay format | Literature data from EUbOPEN Chemogenomic Library | ||
| 12. | ALA5210084 | F | Affinity Phenotypic Cellular interaction (Inhibition of TNF release (in LPS stimulated human macrophages derived from PBMC)) EUB0000265b KDM6A/UTX | Homo sapiens | 1 | assay format | Literature data from EUbOPEN Chemogenomic Library | ||
| 13. | ALA5210576 | B | Affinity Biochemical interaction (AlphaLISA based assay) EUB0000217b KDM6A/UTX | Homo sapiens | 1 | single protein format | Literature data from EUbOPEN Chemogenomic Library | ||
| 14. | ALA5210577 | B | Affinity Biochemical interaction (Mass spectrometry assay) EUB0000265b KDM6A/UTX | Homo sapiens | 1 | single protein format | Literature data from EUbOPEN Chemogenomic Library | ||
| 15. | ALA5216099 | B | Inhibition of KDM6A (unknown origin) expressed in Escherichia coli using Biotin-H3(14-34)K27me3 peptide and measured after 1 hrs by alpha screen assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA5237468 | B | Inhibition of KDM6A (unknown origin ) by TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!