| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2076013 | F | TP_TRANSPORTER: uptake in Xenopus laevis oocytes | Xenopus laevis | 1 | ALA2074516 | cell-based format | TP-search Transporter Database | |
| 2. | ALA2076014 | F | TP_TRANSPORTER: uptake in PEPT1-expressing HRPE cells | 1 | ALA2074516 | cell-based format | TP-search Transporter Database | ||
| 3. | ALA3538386 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30 mins by dual-channel liquid scintillation counting analysis relative to vector control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 4. | ALA3538389 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis relative to vector control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 5. | ALA3540053 | A | Effective permeability of the compound assessed as PepT1-mediated drug uptake in wild type mouse jejunum at 100 uM by HPLC analysis | Mus musculus | 2 | ALA3526020 | single protein format | Scientific Literature | |
| 6. | ALA3540055 | A | Effective permeability of the compound assessed as PepT1-mediated drug uptake in wild type mouse duodenum at 100 uM by HPLC analysis | Mus musculus | 1 | ALA3526020 | single protein format | Scientific Literature | |
| 7. | ALA3540056 | A | Effective permeability of the compound assessed as PepT1-mediated drug uptake in wild type mouse ileum at 100 uM by HPLC analysis | Mus musculus | 1 | ALA3526020 | tissue-based format | Scientific Literature | |
| 8. | ALA3540057 | A | Effective permeability of the compound assessed as PepT1-mediated drug uptake in wild type mouse colon at 100 uM by HPLC analysis | Mus musculus | 1 | ALA3526020 | single protein format | Scientific Literature | |
| 9. | ALA3540998 | A | Activity at mouse recombinant PEPT1 expressed in Pichia pastoris GS115 after 30s by dual-channel liquid scintillation counting analysis | Mus musculus | 1 | ALA3526053 | assay format | Scientific Literature | |
| 10. | ALA3541001 | A | Activity at mouse recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scintillation counting analysis | Mus musculus | 1 | ALA3526053 | assay format | Scientific Literature | |
| 11. | ALA3541260 | A | Ratio of Vmax to Km for mouse recombinant PEPT1 expressed in Pichia pastoris GS115 after 30s by dual-channel liquid scintillation counting analysis | Mus musculus | 1 | ALA3526053 | assay format | Scientific Literature | |
| 12. | ALA3541263 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 13. | ALA3541266 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis in presence of glycine relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 14. | ALA3541269 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis in presence of L-histidine relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 15. | ALA3541272 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis in presence of GlyPro relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 16. | ALA3541275 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis in presence of cefadroxil relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 17. | ALA3534174 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis in presence of SITS relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 18. | ALA3534492 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis in presence of TEA relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 19. | ALA3534495 | A | Drug uptake in Pichia pastoris GS115 expressing mouse recombinant PEPT1 at 5 uM after 30s by dual-channel liquid scintillation counting analysis in presence of elacridar relative to control | Mus musculus | 1 | ALA3526053 | single protein format | Scientific Literature | |
| 20. | ALA3534498 | A | Inhibition of mouse recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation counting analysis | Mus musculus | 1 | ALA3526053 | assay format | Scientific Literature |
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