| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA636543 | B | Selectivity ratio is the antilog of the difference between pA2 values at alpha1- and alpha2- adrenoceptors | Rattus norvegicus | 8 | protein format | Scientific Literature | ||
| 2. | ALA642910 | F | Antagonistic blocking activity at alpha adrenergic receptor by NE induced contractions of the epididymal portion of isolated rat vas deferens at the dose of 20 uM | 36 | tissue-based format | Scientific Literature | |||
| 3. | ALA642911 | B | Binding affinity against Alpha adrenergic receptor using [3H]dihydroergocryptine radioligand in rat brain homogenate | 5 | tissue-based format | Scientific Literature | |||
| 4. | ALA642912 | B | Inhibitory activity against alpha adrenergic receptor | 1 | protein format | Scientific Literature | |||
| 5. | ALA642913 | B | Inhibitory activity against alpha adrenergic receptor in rat | 1 | assay format | Scientific Literature | |||
| 6. | ALA642914 | B | Inhibitory concentration required for displacement of Alpha adrenergic receptor specific ligand, 2-[ [ [(2,6-dimethoxyphenoxy) ethyl]amino]methyl]benzodioxan ([3H]WB-4101) from rat brain cerebral cortical membranes | 6 | cell membrane format | Scientific Literature | |||
| 7. | ALA642915 | F | Antagonism of the pressor response to phenylephrine (10 mg/kg iv) in anesthetized, normotensive rats was determined at a dose range 1-10 mg/kg | 3 | organism-based format | Scientific Literature | |||
| 8. | ALA642916 | F | Antagonism of the pressor response to phenylephrine (10 mg/kg iv) in anesthetized, normotensive rats was determined at a dose range 1-10 mg/kg; Inactive | 1 | organism-based format | Scientific Literature | |||
| 9. | ALA642917 | F | Antagonism of the pressor response to phenylephrine (10 mg/kg iv) in anesthetized, normotensive rats was determined at a dose range 3-30 mg/kg | 1 | organism-based format | Scientific Literature | |||
| 10. | ALA642918 | B | Intrinsic activity against alpha-adrenoceptor in isolated rat tail artery | 3 | protein format | Scientific Literature | |||
| 11. | ALA642919 | B | Intrinsic activity against alpha-adrenoceptor in isolated rat vas deferens | 3 | tissue-based format | Scientific Literature | |||
| 12. | ALA642920 | B | Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranes | 13 | cell membrane format | Scientific Literature | |||
| 13. | ALA642921 | B | Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranes; Inactive | 4 | cell membrane format | Scientific Literature | |||
| 14. | ALA642922 | B | Relative affinity for Alpha adrenergic receptor | 5 | protein format | Scientific Literature | |||
| 15. | ALA642923 | B | Potency(alpha block) relative to labetolol | 5 | protein format | Scientific Literature | |||
| 16. | ALA642924 | F | Evaluated for norepinephrine as agonist. | 1 | assay format | Scientific Literature | |||
| 17. | ALA642925 | F | Evaluated for norepinephrine as agonist. | 1 | assay format | Scientific Literature | |||
| 18. | ALA642926 | F | In vitro postsynaptic antagonist activity against Alpha adrenergic receptor in rat anococcygeus muscle | 5 | tissue-based format | Scientific Literature | |||
| 19. | ALA642927 | F | In vitro presynaptic antagonist activity against Alpha adrenergic receptor in rat vas deferens | 5 | tissue-based format | Scientific Literature | |||
| 20. | ALA640792 | B | In vitro relative blocking action (pA2) of the post-synaptic Alpha adrenergic receptor from rat and rabbit aorta. | 1 | protein format | Scientific Literature |
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